A-196 |
|
Methyltransferase |
SUV420H1/H2 |
A-197, SGC2043 |
No |
07/15 |
A-366 |
|
Methyltransferase |
EHMT2 (G9a), EHMT1 (GLP) |
|
No |
06/13 |
A-395 |
|
WD40 |
EED |
A-395N |
|
07/16 |
BAY-299 |
|
Bromodomains |
BRD1, TAF1 |
BAY-364 |
No |
06/16 |
BAY-598 |
|
Methyltransferase |
SMYD2 |
BAY-369 |
Yes |
04/15 |
BAY-6035 |
|
Methyltransferase |
SMYD3 |
BAY-444 |
|
06/17 |
BAY-850 |
|
Bromodomains |
ATAD2 |
BAY-460 |
|
01/17 |
BAZ2-ICR |
|
Bromodomains |
BAZ2A, BAZ2B |
|
Yes |
05/14 |
BI-9321 |
|
Methyl Lysine Binder |
NSD3 |
BI-9466 |
|
07/18 |
BI-9564 |
|
Bromodomains |
BRD9, BRD7 |
|
Yes |
04/15 |
Bromosporine (BSP) (tool compound) |
|
Bromodomains |
pan-Bromodomain |
|
No |
01/13 |
GSK-J1 use pro-drug GSK-J4 for cell assays |
|
KDM |
KDM6B (JMJD3), KDM6A (UTX), KDM5B (JARID1B) |
GSK-J2 (GSK-J5) |
No |
07/12 |
GSK-LSD1 |
|
KDM |
KDM1A (LSD1) |
|
No |
03/14 |
GSK2801 |
|
Bromodomains |
BAZ2A, BAZ2B |
GSK8573 |
Yes |
12/14 |
GSK343 |
|
Methyltransferase |
EZH2 |
|
No |
08/12 |
GSK4027 |
|
Bromodomains |
KAT2B (PCAF), KAT2A (GCN5) |
GSK4028 |
|
06/17 |
GSK484 |
|
Arginine deiminases |
PAD-4 |
GSK106 |
Yes |
03/15 |
GSK591 |
|
Methyltransferase |
PRMT5 |
SGC2096 |
No |
07/15 |
GSK6853 |
|
Bromodomains |
BRPF1 |
GSK9311 |
Yes |
01/17 |
GSK864 |
|
Dehydrogenase |
Mutant isocitrate dehydrogenase 1 |
GSK990 |
Yes |
11/15 |
GSK8814 |
|
Bromodomains |
ATAD2, ATAD2B |
GSK8815 |
|
01/17 |
Homer |
|
WD40 repeat |
WDR5 |
nc_WDR5 and nc_VHL |
No |
07/21 |
I-BRD9 |
|
Bromodomains |
BRD9 |
|
No |
05/15 |
I-CBP112 |
|
Bromodomains |
CREBBP, EP300 |
|
No |
03/13 |
IOX1 (tool compound) |
|
KDM |
pan-2-OG |
|
No |
01/12 |
IOX2 (requires >>> 1 microM for cell assays) |
|
2OG |
pan-2-OG |
|
No |
02/12 |
JQ1 |
|
Bromodomains |
BRD2, BRD3, BRD4, BRDT (BET) |
(-)-JQ1 |
Yes |
06/10 |
L-Moses |
|
Bromodomains |
KAT2B (PCAF), KAT2A (GCN5) |
D-Moses |
Yes |
10/17 |
LLY-283 |
|
Methyltransferase |
PRMT5 |
LLY-284 |
|
07/16 |
LLY-507 (Multiple Off-target Effects) |
|
Methyltransferase |
SMYD2 |
SGC705 |
No |
11/13 |
LP99 |
|
Bromodomains |
BRD9, BRD7 |
2S,3R-enantiomer |
No |
12/14 |
MRK-740 |
|
Methyltransferase |
PRDM9 |
MRK-740-NC |
|
06/18 |
MRK-952 |
|
|
NUDT5 |
MRK-952-NC |
No |
10/22 |
MRK-990 |
|
|
PRMT9 |
MRK-990-NC |
No |
10/22 |
MS023 |
|
Methyltransferase |
Type I PRMTs (PRMT1,3,4,6,8) |
MS094 |
No |
07/15 |
MS049 |
|
Methyltransferase |
PRMT4 (CARM1), PRMT6 |
MS049N |
No |
06/15 |
NI-57 |
|
Bromodomains |
BRPF1, BRD1 (BRPF2), BRPF3 |
|
No |
12/14 |
NVS-BPTF-1 |
|
Bromodomains |
BPTF (FALZ) |
NVS-BPTF-C |
No |
02/19 |
NVS-CECR2-1 |
|
Bromodomains |
CECR2 |
NVS-CECR2-C |
No |
06/15 |
NVS-MLLT-1 |
|
YEATS |
MLLT1, MLLT3 |
NVS-iMLLT-C |
No |
03/20 |
OF-1 |
|
Bromodomains |
BRPF1, BRD1 (BRPF2), BRPF3 |
|
No |
07/14 |
OICR-9429 |
|
WD40 |
WDR5 |
OICR-0547 |
No |
05/14 |
PFI-1 |
|
Bromodomains |
BRD2, BRD3, BRD4, BRDT (BET) |
|
No |
11/11 |
PFI-2 |
|
Methyltransferase |
SETD7 |
(S)-PFI-2 |
No |
05/13 |
PFI-3 |
|
Bromodomains |
SMARCA2, SMARCA4, PBRM1 (PB1) |
PFI-3oMet |
No |
11/13 |
PFI-4 |
|
Bromodomains |
BRPF1B |
|
No |
12/14 |
PFI-5 |
|
Methyltransferase |
SMYD2 |
PFI-5N |
|
07/17 |
PFI-6 |
|
YEATS |
MLLT1, MLLT3 |
PFI-6N |
No |
06/20 |
PFI-8 |
|
YEATS |
|
PFI-8N |
No |
01/24 |
SGC-CBP30 |
|
Bromodomains |
CREBBP, EP300 |
BDOIA513 |
No |
03/13 |
SGC-SMARCA-BRDVIII |
|
Bromodomains |
SMARCA2/4, PB1(5) |
SGC-BRDVIII-NC |
|
12/20 |
SGC0946 |
|
Methyltransferase |
DOT1L |
SGC0649 |
No |
08/12 |
SGC3027 |
|
Methyltransferase |
PRMT7 |
SGC3027N |
|
03/18 |
SGC6870 |
|
Methyltransferase |
PRMT6 |
SGC6870N |
|
06/19 |
SGC707 |
|
Methyltransferase |
PRMT3 |
XY1 |
No |
06/14 |
SKI-73 |
|
Methyltransferase |
CARM1 (PRMT4) |
SKI-73N |
|
07/17 |
TP-064 |
|
Methyltransferase |
CARM1 (PRMT4) |
TP-064N |
|
06/16 |
TP-238 |
|
Bromodomains |
CECR2, BPTF (FALZ) |
TP-422 |
|
09/18 |
TP-472 |
|
Bromodomains |
BRD9, BRD7 |
TP-472N |
Yes |
06/16 |
UNC0638 |
|
Methyltransferase |
EHMT2 (G9a), EHTM1 (GLP) |
UNC0737 |
No |
06/10 |
UNC0642 |
|
Methyltransferase |
EHMT2 (G9a), EHTM1 (GLP) |
|
Yes |
08/12 |
UNC1215 |
|
Methyl Lysine Binder |
L3MBTL3 |
UNC1079 |
No |
08/12 |
UNC1999 |
|
Methyltransferase |
EZH2 |
UNC2400 |
Yes |
05/13 |
UNC6934 |
|
Methyl Lysine Binder |
NSD2-PWWP1 |
UNC7145 |
|
06/19 |
UNC8732 |
|
Epigenetics |
NSD2 |
UNC8884 |
No |
01/24 |
VinSpinIn |
|
Tudor domains |
Spin1 |
VinSpinIC |
|
09/18 |