A-485
IC50: 0.0026 µM
Pubmed IDs: 28953875

B026

Pubmed IDs: 31910017

Isogarcinol
IC50: 7 µM
Pubmed IDs: 19577000

curcumin derivative 7
IC50: 21 µM
Pubmed IDs: 19577000

Garcinol
IC50: 7 µM
Pubmed IDs: 19577000

LTK-14
IC50: 6 µM
Pubmed IDs: 19577000

curcumin derivative 8
IC50: 33 µM
Pubmed IDs: 19577000

Anacardic acid
IC50: 8.5 µM
Pubmed IDs: 19577000

Lys-coA
IC50: 0.5 µM
Pubmed IDs: 10882143

Nemorosone (activator)
IC50: 5 µM
Pubmed IDs: 20373302

Bowers10_C646
IC50: 1.6 µM
Pubmed IDs: 20534345
Bowers et al. Chemistry and Biology May. 2010

D12-PGJ2
IC50: 0.75 µM
Pubmed IDs: 22141352

NK13650A
IC50: 0.011 µM
Pubmed IDs: 22984806

Windorphen
IC50: 4.2 µM
Pubmed IDs: 24012757

abv15_cmpd700
IC50: 0.011 µM

WO2016044770, WO2016044771, WO2016044777

Diflunisal
IC50: 996 µM
Pubmed IDs: 27244239

Aspirin
IC50: 14000 µM
Pubmed IDs: 27244239

A-485
IC50: 0.0098 µM
Pubmed IDs: 28953875

B026
IC50: 0.0018 µM
Pubmed IDs: 31910017

KAT2B/PCAF


Anacardic acid
IC50: 5 µM
Pubmed IDs: 19577000

Garcinol
IC50: 5 µM
Pubmed IDs: 19577000

Isogarcinol
IC50: 5 µM
Pubmed IDs: 19577000

KAT5/TIP60


MG149
IC50: 74 µM
Pubmed IDs: 22100137

WM-3835
IC50: 0.312 µM
Pubmed IDs: 31827282

wapenaar15_cmpd15
IC50: 37 µM
Pubmed IDs: 26505788

MG149
IC50: 39 µM
Pubmed IDs: 28323055

WM-3835
IC50: 0.03 µM
Pubmed IDs: 31827282

WM-8014
IC50: 0.008 µM
Pubmed IDs: 30069049

WM-1119
IC50: 0.002 µM
Pubmed IDs: 30069049

WM-8014
IC50: 0.008 µM
Pubmed IDs: 31256587

WM-3835
IC50: 0.017 µM
Pubmed IDs: 31827282

WM-8014
IC50: 0.028 µM
Pubmed IDs: 30069049

WM-1119
IC50: 0.002 µM
Pubmed IDs: 30069049
Select All Compounds

A-485

abv15_cmpd700

Anacardic acid

B026

Bowers10_C646

D12-PGJ2

Garcinol

Isogarcinol

LTK-14

Lys-coA

Nemorosone (activator)

NK13650A

Windorphen

WM-1119

WM-3835

WM-8014

WM-8014
Max
IC50
(µM):
 
 

µM