Name In Vivo Activity* Specific Targets Control Post date
VinSpinIn
A chemical probe for the Spin family proteins Spin1 VinSpinIC Sep 2018
TP-238
A chemical probe for CECR2/BPTF bromodomains CECR2/BPTF TP-422 Sep 2018
SGC-GAK-1
A chemical probe for GAK GAK SGC-GAK-1N Feb 2018
SGC-AAK1-1
A dual inhibitor of AAK1 and BMP2K/BIKE AAK1 BMP2K/BIKE SGC-AAK1-1N Feb 2018
BI01383298
A chemical probe for SLC13A5 SLC13A5 BI01372674 Jan 2018
L-Moses
A chemical probe for PCAF and GCN5 Bromodomains yes PCAF, GCN5 D-Moses Oct 2017
BAY-850
A chemical probe for ATAD2A ATAD2 BAY-460 Jan 2017
GSK6853
A chemical probe for BRPF1 yes BRPF1 GSK9311 Jan 2017
TP-472
A BRD9/7 Probe yes BRD9, BRD7 TP-472N Jun 2016
BAY-299
A probe for BRD1 and TAF1 no BRD1, TAF1 BAY-364 Jun 2016
NVS-PAK1-1
A Chemical Probe For PAK1 no PAK1 NVS-PAK1-C Jun 2016
BAY-678
Selective chemical probe for Human Neutrophil Elastase yes Neutrophil Elastase BAY-677 Oct 2015
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