Name In Vivo Activity* Specific Targets Control Post date
NVS-MLLT-1
A Potent and Selective inhibitor of YEATS proteins No MLLT1, MLLT3 NVS-iMLLT-C Mar 2020
SGC6870
A chemical probe for PRMT6 PRMT6 SGC6870N Jun 2019
UNC6934
A chemical probe for NSD2-PWWP1 NSD2-PWWP1 UNC7145 Jun 2019
TP-008
A chemical probe for activin receptor-like kinase (ALK4 and ALK5) No ALK4, ALK5 AI11 May 2019
NVS-BPTF-1
A chemical probe for BPTF No BPTF (FALZ) NVS-BPTF-C Feb 2019
VinSpinIn
A chemical probe for the Spin family proteins Spin1 VinSpinIC Sep 2018
TP-238
A chemical probe for CECR2/BPTF bromodomains CECR2, BPTF (FALZ) TP-422 Sep 2018
DDR-TRK-1
A chemical probe for the DDR and TRK kinase Yes DDR, TRK DDR-TRK-1N Aug 2018
SGC-GAK-1
A chemical probe for GAK GAK SGC-GAK-1N Feb 2018
SGC-AAK1-1
A dual inhibitor of AAK1 and BMP2K/BIKE AAK1 BMP2K/BIKE SGC-AAK1-1N Feb 2018
BI01383298
A chemical probe for SLC13A5 SLC13A5 BI01372674 Jan 2018
L-Moses
A chemical probe for PCAF and GCN5 Bromodomains Yes KAT2B (PCAF), KAT2A (GCN5) D-Moses Oct 2017
PFI-5
A potent inhibitor of SMYD2 with mixed MOA SMYD2 PFI-5N Jul 2017
BAY-850
A chemical probe for ATAD2A ATAD2 BAY-460 Jan 2017
GSK6853
A chemical probe for BRPF1 Yes BRPF1 GSK9311 Jan 2017
TP-472
A BRD9/7 Probe Yes BRD9, BRD7 TP-472N Jun 2016
BAY-299
A probe for BRD1 and TAF1 No BRD1, TAF1 BAY-364 Jun 2016
NVS-PAK1-1
A Chemical Probe For PAK1 No PAK1 NVS-PAK1-C Jun 2016
BAY-678
Selective chemical probe for Human Neutrophil Elastase Yes Neutrophil Elastase BAY-677 Oct 2015
NVS-CECR2-1
A chemical probe for CECR2 No CECR2 NVS-CECR2-C Jun 2015
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