Name |
|
In Vivo Activity* |
Specific Targets |
Control |
Post date |
NVS-MLLT-1 |
A Potent and Selective inhibitor of YEATS proteins |
No |
MLLT1, MLLT3 |
NVS-iMLLT-C |
Mar 2020 |
SGC6870 |
A chemical probe for PRMT6 |
|
PRMT6 |
SGC6870N |
Jun 2019 |
UNC6934 |
A chemical probe for NSD2-PWWP1 |
|
NSD2-PWWP1 |
UNC7145 |
Jun 2019 |
NVS-BPTF-1 |
A chemical probe for BPTF |
No |
BPTF (FALZ) |
NVS-BPTF-C |
Feb 2019 |
VinSpinIn |
A chemical probe for the Spin family proteins |
|
Spin1 |
VinSpinIC |
Sep 2018 |
TP-238 |
A chemical probe for CECR2/BPTF bromodomains |
|
CECR2, BPTF (FALZ) |
TP-422 |
Sep 2018 |
DDR-TRK-1 |
A chemical probe for the DDR and TRK kinase |
Yes |
DDR, TRK |
DDR-TRK-1N |
Aug 2018 |
SGC-GAK-1 |
A chemical probe for GAK |
|
GAK |
SGC-GAK-1N |
Feb 2018 |
SGC-AAK1-1 |
A dual inhibitor of AAK1 and BMP2K/BIKE |
|
AAK1 BMP2K/BIKE |
SGC-AAK1-1N |
Feb 2018 |
BI01383298 |
A chemical probe for SLC13A5 |
|
SLC13A5 |
BI01372674 |
Jan 2018 |
L-Moses |
A chemical probe for PCAF and GCN5 Bromodomains |
Yes |
KAT2B (PCAF), KAT2A (GCN5) |
D-Moses |
Oct 2017 |
PFI-5 |
A potent inhibitor of SMYD2 with mixed MOA |
|
SMYD2 |
PFI-5N |
Jul 2017 |
BAY-850 |
A chemical probe for ATAD2A |
|
ATAD2 |
BAY-460 |
Jan 2017 |
GSK6853 |
A chemical probe for BRPF1 |
Yes |
BRPF1 |
GSK9311 |
Jan 2017 |
TP-472 |
A BRD9/7 Probe |
Yes |
BRD9, BRD7 |
TP-472N |
Jun 2016 |
BAY-299 |
A probe for BRD1 and TAF1 |
No |
BRD1, TAF1 |
BAY-364 |
Jun 2016 |
NVS-PAK1-1 |
A Chemical Probe For PAK1 |
No |
PAK1 |
NVS-PAK1-C |
Jun 2016 |
NVS-CECR2-1 |
A chemical probe for CECR2 |
No |
CECR2 |
NVS-CECR2-C |
Jun 2015 |
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