Selective inhibition of BET bromodomains.

Volume:Pages
468(7327):1067-73
Pubmed id
20871596
Authors

Filippakopoulos P, Qi J, Picaud S, Shen Y, Smith WB, Fedorov O, Morse EM, Keates T, Hickman TT, Felletar I, Philpott M, Munro S, McKeown MR, Wang Y, Christie AL, West N, Cameron MJ, Schwartz B, Heightman TD, La Thangue N, French CA, Wiest O, Kung AL, Knapp S, Bradner JE

DOI
10.1038/nature09504
Journal
Nature
Publication Date
2010-12-23
Year
2010
N Publication Date
PI authors
Validated
Y