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Torres-Fernández LA, Boehm V, Kaufmann J, Becker JP, Garcia-Marquez M, de Bruijn B, Rumińska A, Müller C, Bosco G, Alavinejad N, Lovric L, Bihler JI, Schulte H, Davoodi P, Schöllhorn A, Weihrauch KR, Kaiser L, Ibruli O, Liu F, Androulidaki A, Wobst N, Schmiel M, Valiulis J, Maas L, D'Rozario J, Sakthivelu V, Göbel B, Touet M, Brägelmann J, Höpker K, John F, Wolf J, Knapp S, Quaas A, Cartolano M, von Karstedt S, Beleggia F, Rammensee HG, Gouttefangeas C, Schlößer HA, Riemer AB, Reinhardt HC, Gehring NH, Peifer M, Thomas RK, George J
Mol Cancer. 25(1):. doi: 10.1186/s12943-026-02750-2
Publication date: September 9, 2026
PMID: 42711693
Hiesinger K, Knapp S
J Med Chem. 69(16):19560-19592. doi: 10.1021/acs.jmedchem.6c00996
Publication date: September 1, 2026
PMID: 42679148
Wang X, Mettu A, Herasymenko O, Silva M, Houliston S, Chau I, Ghiabi P, Gibson E, Perveen S, Seitova A, Schapira M, Kireev D
J Chem Inf Model. 66(16):10318-10325. doi: 10.1021/acs.jcim.6c00560
Publication date: August 31, 2026
PMID: 42670858
Zhu WF, Feugray G, Brunst S, Messaoudi H, Yang M, Martinez-Conde N, Krämer A, Weizel L, Ehrler JMH, Kramer JS, Kaiser A, Al-Tarrass M, Pereira T, Valet M, Brunel V, Schubert-Zsilavecz M, Knapp S, Lillich FF, Hernandez-Olmos V, Duflot T, Hiesinger K, Qian H, Proschak A, Bellien J, Proschak E
ACS Chem Biol. 21(8):2053-2067. doi: 10.1021/acschembio.6c00502
Publication date: August 22, 2026
PMID: 42631699
Syphers JL, Wright JA, Kumar A, To N, Elson L, Krämer A, Müller S, Morasch V, Chang A, Young S, Sloan EK, de Nys R, Silva TN, Vrbanac L, Barratt KR, Leeflang J, Hasan ST, Gable RW, Knapp S, Worthley DL, Mukherjee S, Stockton K, Woods SL, Priebbenow DL, Baell JB
J Med Chem. doi: 10.1021/acs.jmedchem.6c00018
Publication date: August 20, 2026
PMID: 42623604
Sanchez-Santos C, Jimenez-Amor A, Martinez-Gonzalez L, Nozal V, Martin-Morales R, Aledavood E, Bausela D, Merrigan K, Diaz-Palacios K, Zhubi R, Knapp S, Garcia-Gonzalo FR, Rodriguez-Cueto C, Gil C, de Lago E, Martinez A
J Med Chem. 69(15):19451-19481. doi: 10.1021/acs.jmedchem.6c01882
Publication date: August 13, 2026
PMID: 42593908
Fraser BJ, Wilson RP, Lac J, Ilyassov O, Seitova A, Li Y, Hutchinson A, Li YY, Loppnau P, Kutera M, Morin GB, Benard F, Arrowsmith CH
J Biol Chem. 113440. doi: 10.1016/j.jbc.2026.113440
Publication date: August 12, 2026
PMID: 42586429
Villagran Suarez A, Hatch KS, Bodrug T, Gai W, Surridge KJ, Moussikhina E, Nguyen KHV, Sanz-Murillo M, Callahan R, Xiong E, Ramos D, Zhu L, Dederer V, Mathea S, Iwasa J, Knapp S, Shokat KM, Reck-Peterson SL, Leschziner AE
Cell. doi: 10.1016/j.cell.2026.07.027
Publication date: August 11, 2026
PMID: 42575089
Lenz C, Saxena K, Knapp S
Methods Mol Biol. 3069:103-124. doi: 10.1007/978-1-0716-5508-5_7
Publication date: August 10, 2026
PMID: 42573692
Frischkorn JM, Riching K, Knapp S, Schwalm MP
Methods Mol Biol. 3069:33-51. doi: 10.1007/978-1-0716-5508-5_3
Publication date: August 10, 2026
PMID: 42573688
Schoppa MQ, Drewry DH
Essays Biochem. doi: 10.1042/EBC20260007
Publication date: July 30, 2026
PMID: 42529985
Willson TM, Merk D
Essays Biochem. doi: 10.1042/EBC20260016
Publication date: July 23, 2026
PMID: 42488934
Madhu P, Benz C, Simonetti L, Winters MJ, Subbanna MS, Kliche J, Gomez-Lucas L, Kotb HM, Krystkowiak I, Segal D, Darling WTP, Larsen-Ledet S, Vieler M, Zupancic A, Konstantinou A, Mihalic F, Varga JK, Pagano L, Lüchow S, Kraemer A, Ellingboe L, Görlitz K, Righetto GL, Kossmann C, Xiong R, Schueler-Furman O, Halabelian L, Santhakumar V, Arrowsmith C, Knapp S, Erdelyi M, Stein A, Vincentelli R, Pryciak PM, Davey NE, Ivarsson Y
bioRxiv. doi: 10.64898/2026.07.03.735260
Publication date: July 17, 2026
PMID: 42465437
Martinov MN, Van Den Bergh A, Jacoby E, Kirov I, Nashev LG, Herasymenko O, Arrowsmith CH, Slater JW, Grell T, Maksimchuk K, Hack MD, Wu Z, Ohadi D, Borrenberghs D, Van Loock M, Mulakala C, Goethals O
J Chem Inf Model. doi: 10.1021/acs.jcim.6c01051
Publication date: July 16, 2026
PMID: 42462159
Joerger AC, Stiewe T
Signal Transduct Target Ther. 11(1):. doi: 10.1038/s41392-026-02830-1
Publication date: July 13, 2026
PMID: 42437754
Liang XJ, Albertini C, Kronenberger T, Shevchenko E, Rasch A, Berger BT, Schwalm M, Berger LM, Krämer A, Serafim RAM, Forster M, Chaikuad A, Bolognesi ML, Müller S, Poso A, Laufer S, Knapp S, Gehringer M
J Med Chem. doi: 10.1021/acs.jmedchem.6c01366
Publication date: July 13, 2026
PMID: 42441922
Anacleto J, Wolf E, Ackloo S, Arrowsmith C, LeBlanc Y, Lento C, Wilson DJ
J Am Chem Soc. doi: 10.1021/jacs.6c03259
Publication date: July 9, 2026
PMID: 42420201
Müller J, Daunke T, Berner N, Bhandare P, Gebhardt A, Hoffmann L, Diebold M, Vogt M, Hofstetter J, Cruz-Garcia Y, Dudvarski-Stankovic N, Schneider K, Adhikari B, Lamer S, Schlosser A, Büchel G, Sos ML, Küster B, Knapp S, Wilhelm S, Wolf E
EMBO Rep. doi: 10.1038/s44319-026-00850-0
Publication date: July 1, 2026
PMID: 42380670
Marsilla J, Welch ML, Siraj J, McElcheran C, Kim JW, Tkachuck D, Kim S, Cho J, Hahn E, Hosni A, Jacinto JC, Kazmierski M, Rey-McIntyre K, Huang SH, Patel T, Tadic T, Bratman S, Hope A, Haibe-Kains B
Phys Imaging Radiat Oncol. 39:101015. doi: 10.1016/j.phro.2026.101015
Publication date: June 30, 2026
PMID: 42376454
Betzholz T, Liu T, Krämer A, Dederer V, Knapp S, Mathea S, Ducho C, Engel M
ChemMedChem. 21(11):e202501007. doi: 10.1002/cmdc.202501007
Publication date: June 18, 2026
PMID: 42313448
Weckesser J, Miletić N, Sivashanmugam SA, Ohmayer U, Steger M, Shashikadze B, Gehrtz P, Unzue Lopez A, Wegener A, Dietz TY, Hammann T, Hartung IV, Elson L, Němec V, Schwalm MP, Adhikari B, Wolf E, Krämer A, Müller S, Daub H, Knapp S
J Med Chem. doi: 10.1021/acs.jmedchem.6c00383
Publication date: June 17, 2026
PMID: 42304961
Ehret TAL, Berger BT, Raig N, Nowotka F, Manik N, Morasch V, Krämer A, Elson L, Matos TL, Müller S, Knapp S, Schwalm MP
ACS Chem Biol. doi: 10.1021/acschembio.6c00410
Publication date: June 15, 2026
PMID: 42287201
Yang D, Wang X, Liu J, Gong Y, Nair P, Sun J, Qian X, Cui J, Zeng H, Dong A, Harding RJ, Burgess-Brown N, Beyett TS, Song D, Krause HM, Diamond ML, Bolhuis DL, Brown NG, Arrowsmith CH, Edwards AM, Halabelian L, Peng H
Proc Natl Acad Sci U S A. 123(25):e2515940123. doi: 10.1073/pnas.2515940123
Publication date: June 5, 2026
PMID: 42247526
Corrionero A, Prendiville N, Cazorla T, Baena-Nuevo M, Sandra R, Camafeita E, Knapp S, Alfonso P
ChemMedChem. 21(11):e70331. doi: 10.1002/cmdc.70331
Publication date: June 4, 2026
PMID: 42236317
Moleón VR, Alende C, Fothouhi M, Bolívar SG, Ayoubi R, Francis V, McPherson PS, Laflamme C
F1000Res. 15:614. doi: 10.12688/f1000research.179367.1
Publication date: June 3, 2026
PMID: 42232299
Edwards M, Amaral A, Carter EM, Arnolds O, Vester K, Thrun A, Wigren E, Homan E, Ribera P, Bentley K, Haraldsson M, Theo-Emegano N, Loppnau P, Szewczyk MM, Cao MA, Barsyte-Lovejoy D, Dittmar N, Hans A, Weber M, Münchow J, Zhu WF, Temme L, Brenker C, Strünker T, Sundström M, Todd MH, Edwards AM, Lesche R, Gileadi O, Tredup C
Hum Reprod. doi: 10.1093/humrep/deag085
Publication date: May 29, 2026
PMID: 42212558
Georgiou EA, Christopoulou K, Kalampaliki AD, Giannopoulou AF, Chatziorfanou E, Bafiti V, Krämer A, Papakyriakou A, Stravopodis DJ, Knapp S, Kostakis IK
ChemMedChem. 21(11):e70324. doi: 10.1002/cmdc.70324
Publication date: May 29, 2026
PMID: 42208521
Greco FA, Abdul Azeez KR, Mitrović M, Sivashanmugam SA, Schwalm MP, Preuss F, Chatterjee D, Morasch V, Mathea S, Hanke T, Müller S, Knapp S
J Med Chem. doi: 10.1021/acs.jmedchem.5c03773
Publication date: May 26, 2026
PMID: 42185966
Bourg S, Place M, Copin C, Chaikuad A, Robert T, Holzmann H, Müller S, Bach S, Ruchaud S, Knapp S, Buron F, Routier S, Bonnet P
Eur J Med Chem. 315:118977. doi: 10.1016/j.ejmech.2026.118977
Publication date: May 24, 2026
PMID: 42176653
Nannini S, Sieffert C, McGown A, Gao XY, Jarvis A, Kostakis GE, Galvacsi A, Kallay C, Moraru R, Baud MG, Mandel S, Balourdas DI, Joerger AC, Orvain C, Peschard S, Nion A, Mellitzer G, Lottiaux S, Spencer J, Gross I, Gaiddon C
J Enzyme Inhib Med Chem. 41(1):2638836. doi: 10.1080/14756366.2026.2638836
Publication date: May 21, 2026
PMID: 42163716
Ferrari ÁJR, Dixit SM, Thibeault J, Garcia M, Houliston S, Ludwig RW, Notin P, Phoumyvong CM, Martell CM, Jung MD, Tsuboyama K, Carter L, Arrowsmith CH, Guttman M, Rocklin GJ
Nature. doi: 10.1038/s41586-026-10465-z
Publication date: May 14, 2026
PMID: 42129553
Klink N, Urban S, Seier JA, Adhikari B, Schwalm MP, Müller J, Dorsch M, Steinbach P, Jung J, Vogt M, Kaschani F, Koch J, Führer S, Kaiser M, Schulze N, Knapp S, Wolf E, Paschen A, Grüner BM, Gersch M
Nat Commun. 17(1):. doi: 10.1038/s41467-026-72295-x
Publication date: May 14, 2026
PMID: 42129197
Andriotti LA, Xavier PLP, Rochetti AL, Qazi TJ, Ferrero AT, de Francisco Strefezzi R, Gomes COMS, Dagli MLZ, Leitão A, Da Silva ER, Muller S, Fukumasu H
Res Vet Sci. 208:106246. doi: 10.1016/j.rvsc.2026.106246
Publication date: May 12, 2026
PMID: 42114276
Ljunggren H, Sokolov A, Ballante F, Fredriksson R, Lagunas-Rangel F, Hauser AS, Knapp S, Jonsson J, Schiöth HB
Br J Pharmacol. doi: 10.1111/bph.70481
Publication date: May 11, 2026
PMID: 42108658
Webb DT, Jones KL, Macabuag N, Bago R, Betts J, Bhattacharyya S, Clifton S, Tinson RAJ, Achara C, Gilbert S, Howell S, Drewry DH, Rogers R, Jones C, Ferguson KR, Bullock AN, Lindsay DM, Kerr WJ, Esmieu W
J Med Chem. doi: 10.1021/acs.jmedchem.6c00714
Publication date: May 4, 2026
PMID: 42076879
Azeez KRA, Saraswati H, Mosler T, Hanke T, Ho-Xuan H, Neder N, Sivashanmugam SA, Heinz M, Schwalm MP, Giuliani G, Rathore R, Kazi R, Kumar R, Mitrovic M, Prieto-Garcia C, Bailey HJ, Mathea S, Hummer G, Đikić I, Müller S, Stolz A, Krause DS, Knapp S
ACS Chem Biol. doi: 10.1021/acschembio.6c00137
Publication date: May 1, 2026
PMID: 42066056
Münick P, Balourdas DI, Funk JS, Yüksel B, Mavridi D, Heftel J, Dreier B, Schaefer JV, Schäfer B, Knapp S, Telatar T, Akgül B, Plückthun A, Stiewe T, Joerger AC, Dötsch V
Proc Natl Acad Sci U S A. 123(18):e2531747123. doi: 10.1073/pnas.2531747123
Publication date: April 28, 2026
PMID: 42048463
Ma J, Huang Y, Zheng T, Wang H, Li B, Liu S, Liu C, Chen X, Min J
Biochem Biophys Res Commun. 819:153815. doi: 10.1016/j.bbrc.2026.153815
Publication date: April 26, 2026
PMID: 42033939
Syphers JL, Wright JA, de Nys R, Silva TN, Vrbanac L, Barratt KR, Leeflang J, Hasan ST, Thomson SF, Kumar A, Krämer A, Lenz C, Gee YS, Chang A, Young S, Sloan EK, Knapp S, Worthley DL, Mukherjee S, Stockton K, Priebbenow DL, Woods SL, Baell JB
Eur J Med Chem. 312:118838. doi: 10.1016/j.ejmech.2026.118838
Publication date: April 25, 2026
PMID: 42030708
Karki R, Vitorino FNL, Searfoss RM, Lempiäinen JK, Arrowsmith CH, Garcia BA
Cell Rep. 45(5):117289. doi: 10.1016/j.celrep.2026.117289
Publication date: April 24, 2026
PMID: 42030158
Robertson KC, Amann SJ, Liu T, Funk AV, Wang X, Grishkovskaya I, Mehmood A, Tabor JR, Norris-Drouin JL, Arrowsmith CH, Collins JL, Miao Y, Emanuele MJ, Haselbach D, James LI, Brown NG
Nat Commun. doi: 10.1038/s41467-026-72235-9
Publication date: April 24, 2026
PMID: 42026065
Hernandez-Olmos V, Patzke JV, Stone CE, Nair RK, Weller K, Sauer F, Endres E, Jamai O, Rachor L, Warmutz CH, Schwalm MP, Mitrovic M, Grenier V, Ehrler JHM, Proschak A, Heering J, Sotriffer C, Mulder MPC, Knapp S, Kisker C, Proschak E
J Med Chem. doi: 10.1021/acs.jmedchem.5c03045
Publication date: April 22, 2026
PMID: 42017948
Emond A, Laflamme C, Therrien M, Liao M, Maios C, Labarre A, Drapeau P, Parker JA
PLoS One. 21(4):e0346613. doi: 10.1371/journal.pone.0346613
Publication date: April 10, 2026
PMID: 41961863
Tessier TM, Maitland MER, Kutera M, Dybas JM, St-Germain J, Arrowsmith CH, Barsyte-Lovejoy D, Zhang W, Raught B, Weitzman MD
Commun Biol. doi: 10.1038/s42003-026-09964-6
Publication date: April 10, 2026
PMID: 41957433
He Y, Bae JSH, Nowak E, Outeiral C, Nissley DA, Tumber A, Berridge G, Salah E, Wang Y, He W, Zhang H, Chen T, Tusk S, Mathea S, Wang YJ, Grassam-Rowe A, Kukura P, Schofield CJ, O'Brien DP, Pierangelini A, Churchill GC, Lanyon-Hogg T, Ke Y, Xu C, Ye T, Watkins H, Ying L, Koschinski A, Solaro RJ, Tan X, Bolla JR, Wang X, Knapp S, Deane CM, Zaccolo M, Nowotny M, Lei M
Cell. doi: 10.1016/j.cell.2026.03.008
Publication date: April 2, 2026
PMID: 41923641
Param NJ, Arceci E, Fiorentino F, Pignata L, Torre D, Gutiérrez-Trejo N, Fong JY, Goy PA, Han BY, Lambona C, Di Bello E, Castiello C, Barone M, Schwarz M, Arrowsmith C, Ito K, Scherle P, Wee DKB, Ndoye S, Tabaglio T, Jeyasekharan AD, Lakshmanan M, Cirilli R, Habisch H, Madl T, Mattevi A, Valente S, Mai A, Guccione E
Sci Adv. 12(13):eaea4059. doi: 10.1126/sciadv.aea4059
Publication date: March 27, 2026
PMID: 41894488
Payliss BJ, Yun HY, Doshi S, Lemak A, Tse YWE, Aprosoff CM, Houliston S, Arrowsmith CH, Wyatt HDM
Nucleic Acids Res. doi: 10.1093/nar/gkag195
Publication date: March 17, 2026
PMID: 41841343
Fanti R, Wolf E, Ikenoue T, Deme JC, Balakrishnan S, Keith BA, Alteen MG, Chandrasekaran R, Yadav M, Bhajiawala R, Ackloo S, Feng J, Pouladi MA, Edwards AM, Wilson DJ, Lea SM, Suga H, Harding RJ
Proc Natl Acad Sci U S A. 123(12):e2520462123. doi: 10.1073/pnas.2520462123
Publication date: March 16, 2026
PMID: 41838909
Knapp S, Weber V, Verheirstraeten M, Sabcheva A, Wright T, Herkens L, Hauser L, Hirschen L, Golzmann A, Lippok B, Krieg S, Ferraris D, Knapp S, Ladurner AG, Rossetti G, Lüscher B, Korn P
Commun Biol. 9(1):. doi: 10.1038/s42003-026-09832-3
Publication date: March 13, 2026
PMID: 41820535
Blas M, Yu C, Aghababazadeh FA, Hoelscher V, Volz M, Morales L, Jarolik K, Dong X, Dobin S, Rantasalo T, Hirvonen T, Pursiheimo JP, Laine N, Homer N, Chamoun C, Pierce W, Organick L, Fehr A, Becich M, Banal JL, Youens K, Tamminen M, Haibe-Kains B, Bedard P
NAR Mol Med. 3(1):ugag011. doi: 10.1093/narmme/ugag011
Publication date: March 9, 2026
PMID: 41797988