Benzodiazepines and benzotriazepines as protein interaction inhibitors targeting bromodomains of the BET family.

Volume:Pages
20(6):1878-86
Pubmed id
22137933
Authors

Filippakopoulos P, Picaud S, Fedorov O, Keller M, Wrobel M, Morgenstern O, Bracher F, Knapp S

DOI
10.1016/j.bmc.2011.10.080
Journal
Bioorg. Med. Chem.
Publication Date
2012-3-15
Year
2012
N Publication Date
PI authors
Validated
Y