Optimization of 3,5-dimethylisoxazole derivatives as potent BET bromodomain ligands.

Pubmed id
23517011
Authors

Hewings DS, Fedorov O, Filippakopoulos P, Martin S, Picaud S, Tumber A, Wells C, Olcina MM, Freeman K, Gill A, Ritchie AJ, Sheppard DW, Russell AJ, Hammond EM, Knapp S, Brennan PE, Conway SJ

DOI
10.1021/jm301588r
Journal
J. Med. Chem.
Publication Date
2013-3-21
Year
2013
N Publication Date
PI authors
Validated
Y