Discovery and Optimization of Small-Molecule Ligands for the CBP/p300 Bromodomains.

Volume:Pages
136(26):9308-19
Pubmed id
24946055
Authors

Hay DA, Fedorov O, Martin S, Singleton DC, Tallant C, Wells C, Picaud S, Philpott M, Monteiro OP, Rogers CM, Conway SJ, Rooney TP, Tumber A, Yapp C, Filippakopoulos P, Bunnage ME, Müller S, Knapp S, Schofield CJ, Brennan PE

DOI
10.1021/ja412434f
Journal
J. Am. Chem. Soc.
Publication Date
2014-7-2
Year
2014
N Publication Date
PI authors
Validated
Y