A unique inhibitor binding site in ERK1/2 is associated with slow binding kinetics.

Site
Pubmed id
25195011
Authors

Chaikuad A, M C Tacconi E, Zimmer J, Liang Y, Gray NS, Tarsounas M, Knapp S

DOI
10.1038/nchembio.1629
Journal
Nat. Chem. Biol.
Publication Date
2014-9-7
Year
2014
N Publication Date
PI authors
Validated
Y