The 9H-purine scaffold reveals induced-fit pocket plasticity of the BRD9 bromodomain.

Site
Pubmed id
25703523
Authors

Picaud S, Strocchia M, Terracciano S, Lauro G, Méndez J, Daniels DL, Riccio R, Bifulco G, Bruno I, Filippakopoulos P

DOI
10.1021/jm501893k
Journal
J. Med. Chem.
Publication Date
2015-2-22
Year
2015
N Publication Date
Validated
Y