Generation of a selective small molecule inhibitor of the CBP/p300 bromodomain for leukemia therapy.

Pubmed id
26552700
Authors

Picaud S, Fedorov O, Thanasopoulou A, Leonards K, Jones K, Meier J, Olzscha H, Monteiro O, Martin S, Philpott M, Tumber A, Filippakopoulos P, Yapp C, Wells C, Hing Che K, Bannister A, Robson S, Kumar U, Parr N, Lee K, Lugo D, Jeffrey P, Taylor S, Vecellio ML, Bountra C, Brennan P, O'Mahony A, Velichko S, Muller S, Hay D, Daniels DL, Urh M, La Thangue NB, Kouzarides T, Prinjha R, Schwaller J, Knapp S

DOI
10.1158/0008-5472.CAN-15-0236
Journal
Cancer Res.
Publication Date
2015-11-9
Year
2015
N Publication Date
PI authors
Validated
Y