Structure-based identification of inhibitory fragments targeting the p300/CBP-associated factor bromodomain.

Pubmed id
26731131
Authors

Chaikuad A, Lang S, Brennan PE, Temperini C, Fedorov O, Hollander J, Nachane R, Abell C, Müller S, Siegal G, Knapp S

DOI
10.1021/acs.jmedchem.5b01719
Journal
J. Med. Chem.
Publication Date
2016-1-5
Year
2016
N Publication Date
PI authors
Validated
Y