Exploring Selective Inhibition of the First Bromodomain of the Human Bromodomain and Extra-terminal Domain (BET) Proteins.

Site
Pubmed id
26735842
Authors

Raux B, Voitovich Y, Derviaux C, Lugari A, Rebuffet E, Milhas S, Priet S, Roux T, Trinquet E, Guillemot JC, Knapp S, Brunel JM, Fedorov AY, Collette Y, Roche P, Betzi S, Combes S, Morelli X

DOI
10.1021/acs.jmedchem.5b01708
Journal
J. Med. Chem.
Publication Date
2016-1-6
Year
2016
N Publication Date
PI authors
Validated
Y