Identification of a chemical probe for family VIII bromodomains through optimization of a fragment hit.

Pubmed id
27115555
Authors

Gerstenberger BS, Trzupek JD, Tallant C, Fedorov O, Filippakopoulos P, Brennan PE, Fedele V, Martin S, Picaud S, Rogers CM, Parikh MD, Taylor A, Samas BM, O'Mahony A, Berg EL, Pallares G, Torrey AV, Treiber DK, Samardjiev IJ, Nasipak BT, Padilla-Benavides T, Wu Q, Imbalzano AN, Nickerson JA, Bunnage ME, Müller S, Knapp S, Owen DR

DOI
10.1021/acs.jmedchem.6b00012
Journal
J. Med. Chem.
Publication Date
2016-4-26
Year
2016
N Publication Date
PI authors
Validated
Y