Covalent targeting of remote cysteine residues to develop CDK12 and CDK13 inhibitors.

Site
Pubmed id
27571479
Authors

Zhang T, Kwiatkowski N, Olson CM, Dixon-Clarke SE, Abraham BJ, Greifenberg AK, Ficarro SB, Elkins JM, Liang Y, Hannett NM, Manz T, Hao M, Bartkowiak B, Greenleaf AL, Marto JA, Geyer M, Bullock AN, Young RA, Gray NS

DOI
10.1038/nchembio.2166
Journal
Nat. Chem. Biol.
Publication Date
2016-8-29
Year
2016
N Publication Date
Validated
Y