An Unusual Binding Model of the Methyl 9-Anilinothiazolo[5,4-f] quinazoline-2-carbimidates (EHT 1610 and EHT 5372) Confers High Selectivity for Dual-specificity Tyrosine Phosphorylation-Regulated Kinases.

Site
Pubmed id
27766861
Authors

Chaikuad A, Diharce J, Schröder M, Foucourt A, Leblond B, Casagrande AS, Desire L, Bonnet P, Knapp S, Besson T

DOI
10.1021/acs.jmedchem.6b01083
Journal
J. Med. Chem.
Publication Date
2016-10-21
Year
2016
N Publication Date
PI authors
Validated
Y