Turning a Substrate Peptide into a Potent Inhibitor for the Histone Methyltransferase SETD8.

Volume:Pages
7(12):1102-1106
Site
Pubmed id
27994746
Authors

Judge RA, Zhu H, Upadhyay AK, Bodelle PM, Hutchins CW, Torrent M, Marin VL, Yu W, Vedadi M, Li F, Brown PJ, Pappano WN, Sun C, Petros AM

DOI
10.1021/acsmedchemlett.6b00303
Journal
ACS Med Chem Lett
Publication Date
2016-12-8
Year
2016
N Publication Date
Validated
Y