Benzo-isoquinoline-diones As Potent and Selective Inhibitors of BRPF2 and TAF1/TAF1L Bromodomains.

Pubmed id
28402630
Authors

Bouché L, Christ CD, Siegel S, Fernández-Montalván AE, Holton SJ, Fedorov O, Ter Laak A, Sugawara T, Stöckigt D, Tallant C, Bennett JM, Monteiro OP, Díaz-Sáez L, Siejka P, Meier J, Puetter V, Weiske J, Müller S, Huber KV, Hartung IV, Haendler B

DOI
10.1021/acs.jmedchem.7b00306
Journal
J. Med. Chem.
Publication Date
2017-4-12
Year
2017
N Publication Date
Validated
Y