Discovery of a highly selective cell-active inhibitor of KDM2/7.

Pubmed id
28976073
Authors

Gerken P, Wolstenhulme J, Tumber A, Hatch S, Zhang Y, Müller S, Chandler S, Mair B, Li F, Nijman S, Konietzny R, Szommer T, Yapp C, Fedorov O, Benesch J, Vedadi M, Kessler B, Kawamura A, Brennan P, Smith MD

DOI
10.1002/anie.201706788
Journal
Angew. Chem. Int. Ed. Engl.
Publication Date
2017-10-4
Year
2017
N Publication Date
Validated
Y