GW779439X and its pyrazolopyridazine derivatives inhibit the serine/threonine kinase Stk1 and act as antibiotic adjuvants against β-lactam-resistant Staphylococcus aureus.

Site
Pubmed id
30059625
Authors

Schaenzer AJ, Wlodarchak N, Drewry D, Zuercher WJ, Rose WE, Ferrer CA, Sauer JD, Striker R

DOI
10.1021/acsinfecdis.8b00136
Journal
ACS Infect Dis
Publication Date
2018-7-30
Year
2018
N Publication Date
PI authors
Validated
Y