Rapid covalent-probe discovery by electrophile-fragment screening.

Site
Pubmed id
31060360
Authors

Resnick E, Bradley A, Gan J, Douangamath A, Krojer T, Sethi R, Geurink PP, Aimon A, Amitai G, Bellini D, Bennett J, Fairhead M, Fedorov O, Gabizon R, Gan J, Guo J, Plotnikov A, Reznik N, Ruda GF, Díaz-Sáez L, Straub VM, Szommer T, Velupillai S, Zaidman D, Zhang Y, Coker AR, Dowson CG, Barr H, Wang C, Huber KVM, Brennan PE, Ovaa H, von Delft F, London N

DOI
10.1021/jacs.9b02822
Journal
J. Am. Chem. Soc.
Publication Date
2019-5-7
Year
2019
N Publication Date
Validated
Y