Identification and characterization of the first fragment hits for SETDB1 Tudor domain.

Site
Pubmed id
31327677
Authors

Mader P, Mendoza-Sanchez R, Iqbal A, Dong A, Dobrovetsky E, Corless VB, Liew SK, Houliston SR, De Freitas RF, Smil D, Sena CCD, Kennedy S, Diaz DB, Wu H, Dombrovski L, Allali-Hassani A, Min J, Schapira M, Vedadi M, Brown PJ, Santhakumar V, Yudin AK, Arrowsmith CH

DOI
10.1016/j.bmc.2019.07.020
Journal
Bioorg. Med. Chem.
Publication Date
2019-7-12
Year
2019
N Publication Date
PI authors
Validated
Y