A Chemical Probe for Dark Kinase STK17B Derives Its Potency and High Selectivity through a Unique P-Loop Conformation.

Site
Pubmed id
33215924
Authors

Picado A, Chaikuad A, Wells CI, Shrestha S, Zuercher WJ, Pickett JE, Kwarcinski FE, Sinha P, de Silva CS, Zutshi R, Liu S, Kannan N, Knapp S, Drewry DH, Willson TM

DOI
10.1021/acs.jmedchem.0c01174
Journal
J Med Chem
Publication Date
2020-11-20
Year
2020
N Publication Date
PI authors
Validated
Y