Structure-kinetic relationship reveals the mechanism of selectivity of FAK inhibitors over PYK2.

Pubmed id
33497606
Authors

Berger BT, Amaral M, Kokh DB, Nunes-Alves A, Musil D, Heinrich T, Schröder M, Neil R, Wang J, Navratilova I, Bomke J, Elkins JM, Müller S, Frech M, Wade RC, Knapp S

DOI
10.1016/j.chembiol.2021.01.003
Journal
Cell Chem Biol
Publication Date
2021-1-21
Year
2021
N Publication Date
PI authors
Validated
Y