Structure-Guided Development of Small-Molecule PRC2 Inhibitors Targeting EZH2-EED Interaction.

Site
Pubmed id
34077206
Authors

Du D, Xu D, Zhu L, Stazi G, Zwergel C, Liu Y, Luo Z, Li Y, Zhang Y, Zhu K, Ding Y, Liu J, Fan S, Zhao K, Zhang N, Kong X, Jiang H, Chen K, Zhao K, Valente S, Min J, Duan W, Luo C

DOI
10.1021/acs.jmedchem.0c02261
Journal
J Med Chem
Publication Date
2021-6-2
Year
2021
N Publication Date
Validated
Y