Demonstration of the utility of DOS-derived fragment libraries for rapid hit derivatisation in a multidirectional fashion.

Volume:Pages
11(39):10792-10801
Site
Pubmed id
34094333
Authors

Kidd SL, Fowler E, Reinhardt T, Compton T, Mateu N, Newman H, Bellini D, Talon R, McLoughlin J, Krojer T, Aimon A, Bradley A, Fairhead M, Brear P, Díaz-Sáez L, McAuley K, Sore HF, Madin A, O'Donovan DH, Huber KVM, Hyvönen M, von Delft F, Dowson CG, Spring DR

DOI
10.1039/d0sc01232g
Journal
Chem Sci
Publication Date
2020-5-14
Year
2020
N Publication Date
Validated
Y