Development of the First Covalent Monopolar Spindle Kinase 1 (MPS1/TTK) Inhibitor.

Pubmed id
35167750
Authors

M Serafim RA, da Silva Santiago A, Schwalm MP, Hu Z, Dos Reis CV, Takarada JE, Mezzomo P, Massirer KB, Kudolo M, Gerstenecker S, Chaikuad A, Zender L, Knapp S, Laufer S, Couñago RM, Gehringer M

DOI
10.1021/acs.jmedchem.1c01165
Journal
J Med Chem
Publication Date
2022-2-15
Year
2022
N Publication Date
PI authors
Validated
Y