Identification of Novel 2,4,5-Trisubstituted Pyrimidines as Potent Dual Inhibitors of Plasmodial PfGSK3/PfPK6 with Activity against Blood Stage Parasites In Vitro.

Site
Pubmed id
36166733
Authors

Galal KA, Truong A, Kwarcinski F, de Silva C, Avalani K, Havener TM, Chirgwin ME, Merten E, Ong HW, Willis C, Abdelwaly A, Helal MA, Derbyshire ER, Zutshi R, Drewry DH

DOI
10.1021/acs.jmedchem.2c00996
Journal
J Med Chem
Publication Date
2022-9-27
Year
2022
N Publication Date
PI authors
Validated
Y