Development of Highly Potent and Selective Covalent FGFR4 Inhibitors Based on SNAr Electrophiles.

Site
Pubmed id
38604131
Authors

Schwarz M, Kurkunov M, Wittlinger F, Rudalska R, Wang G, Schwalm MP, Rasch A, Wagner B, Laufer SA, Knapp S, Dauch D, Gehringer M

DOI
10.1021/acs.jmedchem.3c02483
Journal
J Med Chem
Publication Date
2024-4-11
Year
2024
N Publication Date
PI authors
Validated
Y