Crystal structure of the first bromodomain of human BRD4 in complex with a tetrahydroquinoline analogue

Protein: BRD4
PDB ID: 5N2M
Deposition Date: Tuesday 7th February 2017
Authors: Tallant, C., Slavish, P.J., Siejka, P., Bharatham, N., Shadrick, W.R., Chai, S., Young, B.M., Boyd, V.A., Heroven, C., Wiggers, H.J., Picaud, S., Fedorov, O., Krojer, T., Chen, T., Lee, R.E., Guy, R.K., Shelat, A.A., von Delft, F., Arrowsmith, C.H., Edwards, A.M., Bountra, C., Knapp, S.