Discovery of a Potent Class I Protein Arginine Methyltransferase Fragment Inhibitor.

Site
Pubmed id
26824386
Authors

Ferreira de Freitas R, Eram MS, Szewczyk MM, Steuber H, Smil D, Wu H, Li F, Senisterra G, Dong A, Brown PJ, Hitchcock M, Moosmayer D, Stegmann CM, Egner U, Arrowsmith C, Barsyte-Lovejoy D, Vedadi M, Schapira M

DOI
10.1021/acs.jmedchem.5b01772
Journal
J. Med. Chem.
Publication Date
2016-1-29
Year
2016
N Publication Date
Validated
Y