Discovery of potent Plasmodium falciparum protein kinase 6 (PfPK6) inhibitors with a type II inhibitor pharmacophore.

Volume:Pages
249:115043
Site
Pubmed id
36736152
Authors

Ong HW, Truong A, Kwarcinski F, de Silva C, Avalani K, Havener TM, Chirgwin M, Galal KA, Willis C, Krämer A, Liu S, Knapp S, Derbyshire ER, Zutshi R, Drewry DH

DOI
10.1016/j.ejmech.2022.115043
Journal
Eur J Med Chem
Publication Date
2022-12-30
Year
2022
N Publication Date
PI authors
Validated
Y