Discovery of a Potent and Selective Targeted NSD2 Degrader for the Reduction of H3K36me2.

Site
Pubmed id
36976643
Authors

Hanley RP, Nie DY, Tabor JR, Li F, Sobh A, Xu C, Barker NK, Dilworth D, Hajian T, Gibson E, Szewczyk MM, Brown PJ, Barsyte-Lovejoy D, Herring LE, Wang GG, Licht JD, Vedadi M, Arrowsmith CH, James LI

DOI
10.1021/jacs.3c01421
Journal
J Am Chem Soc
Publication Date
2023-3-28
Year
2023
N Publication Date
Validated
Y