Development of HC-258, a Covalent Acrylamide TEAD Inhibitor That Reduces Gene Expression and Cell Migration.

Volume:Pages
14(12):1746-1753
Site
Pubmed id
38116405
Authors

Fnaiche A, Chan HC, Paquin A, González Suárez N, Vu V, Li F, Allali-Hassani A, Cao MA, Szewczyk MM, Bolotokova A, Allemand F, Gelin M, Barsyte-Lovejoy D, Santhakumar V, Vedadi M, Guichou JF, Annabi B, Gagnon A

DOI
10.1021/acsmedchemlett.3c00386
Journal
ACS Med Chem Lett
Publication Date
2023-12-14
Year
2023
N Publication Date
PI authors
Validated
Y