Druggability analysis and structural classification of bromodomain acetyl-lysine binding sites. Read more about Druggability analysis and structural classification of bromodomain acetyl-lysine binding sites.
An allosteric inhibitor of protein arginine methyltransferase 3. Read more about An allosteric inhibitor of protein arginine methyltransferase 3.
Structure and mechanism of human UDP-xylose synthase: evidence for a promoting role of sugar ring distortion in a three-step catalytic conversion of UDP-glucuronic acid. Read more about Structure and mechanism of human UDP-xylose synthase: evidence for a promoting role of sugar ring distortion in a three-step catalytic conversion of UDP-glucuronic acid.
Targeting kinases for the treatment of inflammatory diseases. Read more about Targeting kinases for the treatment of inflammatory diseases.
Discovery of ligands for ADP-ribosyltransferases via docking-based virtual screening. Read more about Discovery of ligands for ADP-ribosyltransferases via docking-based virtual screening.
A selective jumonji H3K27 demethylase inhibitor modulates the proinflammatory macrophage response. Read more about A selective jumonji H3K27 demethylase inhibitor modulates the proinflammatory macrophage response.
Small-molecule inhibition of BRDT for male contraception. Read more about Small-molecule inhibition of BRDT for male contraception.
Structural determination of the phosphorylation domain of the ryanodine receptor. Read more about Structural determination of the phosphorylation domain of the ryanodine receptor.
Structural basis for ASPP2 recognition by the tumor suppressor p73. Read more about Structural basis for ASPP2 recognition by the tumor suppressor p73.
Fragment screening of cyclin G-associated kinase by weak affinity chromatography. Read more about Fragment screening of cyclin G-associated kinase by weak affinity chromatography.
