Discovery of ligands for ADP-ribosyltransferases via docking-based virtual screening. Read more about Discovery of ligands for ADP-ribosyltransferases via docking-based virtual screening.
A selective jumonji H3K27 demethylase inhibitor modulates the proinflammatory macrophage response. Read more about A selective jumonji H3K27 demethylase inhibitor modulates the proinflammatory macrophage response.
Small-molecule inhibition of BRDT for male contraception. Read more about Small-molecule inhibition of BRDT for male contraception.
Structural determination of the phosphorylation domain of the ryanodine receptor. Read more about Structural determination of the phosphorylation domain of the ryanodine receptor.
Structural basis for ASPP2 recognition by the tumor suppressor p73. Read more about Structural basis for ASPP2 recognition by the tumor suppressor p73.
Fragment screening of cyclin G-associated kinase by weak affinity chromatography. Read more about Fragment screening of cyclin G-associated kinase by weak affinity chromatography.
Crystal structure of human aurora B in complex with INCENP and VX-680. Read more about Crystal structure of human aurora B in complex with INCENP and VX-680.
Pyruvate kinase M2 activators promote tetramer formation and suppress tumorigenesis. Read more about Pyruvate kinase M2 activators promote tetramer formation and suppress tumorigenesis.
Progress in the Development and Application of Small Molecule Inhibitors of Bromodomain-Acetyl-lysine Interactions. Read more about Progress in the Development and Application of Small Molecule Inhibitors of Bromodomain-Acetyl-lysine Interactions.
Structures of human DPP7 reveal the molecular basis of specific inhibition and the architectural diversity of proline-specific peptidases. Read more about Structures of human DPP7 reveal the molecular basis of specific inhibition and the architectural diversity of proline-specific peptidases.
