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Tjaden A, Knapp S, Müller S
Methods Mol Biol. 2706:59-73. doi: 10.1007/978-1-0716-3397-7_5
Publication date: August 10, 2023
PMID: 37558941
Elson L, Tjaden A, Knapp S, Müller S
Methods Mol Biol. 2706:75-88. doi: 10.1007/978-1-0716-3397-7_6
Publication date: August 10, 2023
PMID: 37558942
Wells CI, Drewry DH
Methods Mol Biol. 2706:11-24. doi: 10.1007/978-1-0716-3397-7_2
Publication date: August 10, 2023
PMID: 37558938
Bhattacharya D, Shi Ming Li A, Paul B, Ghosh Dastidar U, Santhakumar V, Sarkar D, Chau I, Li F, Ghosh T, Vedadi M, Talukdar A
Eur J Med Chem. 260:115713. doi: 10.1016/j.ejmech.2023.115713
Publication date: August 10, 2023
PMID: 37597437
Ramachandran S, Szewczyk M, Barghout SH, Ciulli A, Barsyte-Lovejoy D, Vu V
Methods Mol Biol. 2706:149-165. doi: 10.1007/978-1-0716-3397-7_11
Publication date: August 10, 2023
PMID: 37558947
Szewczyk MM, Owens DDG, Barsyte-Lovejoy D
Methods Mol Biol. 2706:137-148. doi: 10.1007/978-1-0716-3397-7_10
Publication date: August 10, 2023
PMID: 37558946
Němec V, Knapp S
Methods Mol Biol. 2706:51-58. doi: 10.1007/978-1-0716-3397-7_4
Publication date: August 10, 2023
PMID: 37558940
Uguen M, Deng Y, Li F, Shell DJ, Norris-Drouin JL, Stashko MA, Ackloo S, Arrowsmith CH, James LI, Liu P, Pearce KH, Frye SV
ACS Chem Biol. doi: 10.1021/acschembio.3c00280
Publication date: August 9, 2023
PMID: 37556795
Ayoubi R, Fotouhi M, Southern K, Bhajiawala R, Fanti R, Prinos P, McPherson PS, Laflamme C
F1000Res. 12:308. doi: 10.12688/f1000research.131333.1
Publication date: August 7, 2023
PMID: 37545650
Harding RJ, Franzoni I, Mann MK, Szewczyk MM, Mirabi B, Ferreira de Freitas R, Owens DDG, Ackloo S, Scheremetjew A, Juarez-Ornelas KA, Sanichar R, Baker RJ, Dank C, Brown PJ, Barsyte-Lovejoy D, Santhakumar V, Schapira M, Lautens M, Arrowsmith CH
J Med Chem. doi: 10.1021/acs.jmedchem.3c00314
Publication date: July 27, 2023
PMID: 37499118
Tilley L, Xie S, Wang Y, Morton C, Metcalfe R, Dogovski C, Pasaje CF, Dunn E, Luth M, Kumpornsin K, Istvan E, Park J, Fairhurst K, Yeo T, Yildirim O, Bhebhe M, Klug D, Rutledge P, Godoy L, Dey S, De Souza M, Siqueira-Neto J, Ketprasit N, Du Y, Amini M, Shami G, Nie S, Williamson N, Jana G, Maity B, Thomson P, Foley T, Loesbanluechai D, Puhalovich T, Tan D, Niles J, Han BW, Goldberg D, Burrows J, Fidock D, Lee M, Winzeler E, Griffin M, Todd M
Res Sq. doi: 10.21203/rs.3.rs-3198291/v1
Publication date: July 27, 2023
PMID: 37546892
Harding RJ, Bermudez P, Bernier A, Beauvais M, Bellec P, Hill S, Karakuzu A, Knoppers BM, Pavlidis P, Poline JB, Roskams J, Stikov N, Stone J, Strother S, Evans AC
PLoS Comput Biol. 19(7):e1011230. doi: 10.1371/journal.pcbi.1011230
Publication date: July 27, 2023
PMID: 37498959
Chauhan C, Kraemer A, Knapp S, Windheim M, Kotlyarov A, Menon MB, Gaestel M
Cell Death Discov. 9(1):262. doi: 10.1038/s41420-023-01576-x
Publication date: July 26, 2023
PMID: 37495567
Castano A, Silvestre M, Wells CI, Sanderson JL, Ferrer CA, Ong HW, Lang Y, Richardson W, Silvaroli JA, Bashore FM, Smith JL, Genereux IM, Dempster K, Drewry DH, Pabla NS, Bullock AN, Benke TA, Ultanir S, Axtman AD
Elife. 12:. doi: 10.7554/eLife.88206
Publication date: July 25, 2023
PMID: 37490324
Deau E, Lindberg MF, Miege F, Roche D, George N, George P, Krämer A, Knapp S, Meijer L
J Med Chem. doi: 10.1021/acs.jmedchem.3c00884
Publication date: July 24, 2023
PMID: 37487467
Arifi S, Marschner JA, Pollinger J, Isigkeit L, Heitel P, Kaiser A, Obeser L, Höfner G, Proschak E, Knapp S, Chaikuad A, Heering J, Merk D
J Am Chem Soc. doi: 10.1021/jacs.3c03417
Publication date: June 29, 2023
PMID: 37385602
Negoita F, Addinsall AB, Hellberg K, Bringas CF, Hafen PS, Sermersheim TJ, Agerholm M, Lewis CTA, Ahwazi D, Ling NXY, Larsen JK, Deshmukh AS, Hossain MA, Oakhill JS, Ochala J, Brault JJ, Sankar U, Drewry DH, Scott JW, Witczak CA, Sakamoto K
Mol Metab. 101761. doi: 10.1016/j.molmet.2023.101761
Publication date: June 26, 2023
PMID: 37380024
Kimani SW, Owen J, Green SR, Li F, Li Y, Dong A, Brown PJ, Ackloo S, Kuter D, Yang C, MacAskill M, MacKinnon SS, Arrowsmith CH, Schapira M, Shahani V, Halabelian L
J Chem Inf Model. doi: 10.1021/acs.jcim.3c00082
Publication date: June 23, 2023
PMID: 37350740
Ackloo S, Antolin AA, Bartolome JM, Beck H, Bullock A, Betz UAK, Böttcher J, Brown PJ, Chaturvedi M, Crisp A, Daniels D, Dreher J, Edfeldt K, Edwards AM, Egner U, Elkins J, Fischer C, Glendorf T, Goldberg S, Hartung IV, Hillisch A, Homan E, Knapp S, Köster M, Krämer O, Llaveria J, Lessel U, Lindemann S, Linderoth L, Matsui H, Michel M, Montel F, Mueller-Fahrnow A, Müller S, Owen DR, Saikatendu KS, Santhakumar V, Sanderson W, Scholten C, Schapira M, Sharma S, Shireman B, Sundström M, Todd MH, Tredup C, Venable J, Willson TM, Arrowsmith CH
RSC Med Chem. 14(6):1002-1011. doi: 10.1039/d2md00441k
Publication date: June 22, 2023
PMID: 37360399
Alteen MG, Deme JC, Alvarez CP, Loppnau P, Hutchinson A, Seitova A, Chandrasekaran R, Silva Ramos E, Secker C, Alqazzaz M, Wanker EE, Lea SM, Arrowsmith CH, Harding RJ
Structure. doi: 10.1016/j.str.2023.06.002
Publication date: June 20, 2023
PMID: 37390814
Schwalm MP, Krämer A, Dölle A, Weckesser J, Yu X, Jin J, Saxena K, Knapp S
Cell Chem Biol. doi: 10.1016/j.chembiol.2023.06.002
Publication date: June 20, 2023
PMID: 37354907
Singh I, Li F, Fink EA, Chau I, Li A, Rodriguez-Hernández A, Glenn I, Zapatero-Belinchón FJ, Rodriguez ML, Devkota K, Deng Z, White K, Wan X, Tolmachova NA, Moroz YS, Kaniskan HÜ, Ott M, GarcÃa-Sastre A, Jin J, Fujimori DG, Irwin JJ, Vedadi M, Shoichet BK
J Med Chem. doi: 10.1021/acs.jmedchem.2c02120
Publication date: June 9, 2023
PMID: 37294077
Amrhein JA, Wang G, Berger BT, Berger LM, Kalampaliki AD, Krämer A, Knapp S, Hanke T
ACS Med Chem Lett. 14(6):833-840. doi: 10.1021/acsmedchemlett.3c00127
Publication date: June 8, 2023
PMID: 37312836
Ni X, Joerger AC, Chaikuad A, Knapp S
Open Biol. 13(5):230031. doi: 10.1098/rsob.230031
Publication date: May 31, 2023
PMID: 37253421
Novak L, Petrosino M, Pasquo A, Chaikuad A, Chiaraluce R, Knapp S, Consalvi V
Cancers (Basel). 15(11):. doi: 10.3390/cancers15112938
Publication date: May 26, 2023
PMID: 37296900
Marcelino TP, Fala AM, da Silva MM, Souza-Melo N, Malvezzi AM, Klippel AH, Zoltner M, Padilla-Mejia N, Kosto S, Field MC, Burle Caldas GA, Teixeira SMR, Couñago RM, Massirer KB, Schenkman S
J Biol Chem. 104857. doi: 10.1016/j.jbc.2023.104857
Publication date: May 23, 2023
PMID: 37230387
Axtman AD, Brennan PE, Frappier-Brinton T, Betarbet R, Carter GW, Fu H, Gileadi O, Greenwood AK, Leal K, Longo FM, Mangravite LM, Edwards AM, Levey AI
Alzheimers Dement (N Y). 9(2):e12394. doi: 10.1002/trc2.12394
Publication date: May 22, 2023
PMID: 37215505
Choi JY, Noguchi Y, Alburger JM, Bayle S, Chung E, Grant W, Chaikuad A, Knapp S, Duckett DR, Roush WR
J Med Chem. doi: 10.1021/acs.jmedchem.2c01180
Publication date: May 19, 2023
PMID: 37204207
Nam J, Schirmer AU, Loh C, Drewry DH, Macias E
Cancers (Basel). 15(10):. doi: 10.3390/cancers15102817
Publication date: May 18, 2023
PMID: 37345153
Scantlebury J, Vost L, Carbery A, Hadfield TE, Turnbull OM, Brown N, Chenthamarakshan V, Das P, Grosjean H, von Delft F, Deane CM
J Chem Inf Model. doi: 10.1021/acs.jcim.3c00322
Publication date: May 11, 2023
PMID: 37166179
Cunha MR, Catta-Preta CMC, Takarada JE, Moreira GA, Massirer KB, Couñago RM
J Biol Chem. 104807. doi: 10.1016/j.jbc.2023.104807
Publication date: May 10, 2023
PMID: 37172730
Durcan TM, Axtman AD
Front Cell Neurosci. 17:1196543. doi: 10.3389/fncel.2023.1196543
Publication date: May 1, 2023
PMID: 37124399
Hargittay B, Mineev KS, Richter C, Sreeramulu S, Jonker HRA, Saxena K, Schwalbe H
Biomol NMR Assign. doi: 10.1007/s12104-023-10132-8
Publication date: April 29, 2023
PMID: 37118562
Ong HW, Liang Y, Richardson W, Lowry ER, Wells CI, Chen X, Silvestre M, Dempster K, Silvaroli JA, Smith JL, Wichterle H, Pabla NS, Ultanir SK, Bullock AN, Drewry DH, Axtman AD
ACS Chem Neurosci. doi: 10.1021/acschemneuro.3c00135
Publication date: April 21, 2023
PMID: 37084253
Liu K, Zhang J, Xiao Y, Yang A, Song X, Li Y, Chen Y, Hughes TR, Min J
J Biol Chem. 104734. doi: 10.1016/j.jbc.2023.104734
Publication date: April 20, 2023
PMID: 37086783
Bashore FM, Marquez AB, Chaikuad A, Howell S, Dunn AS, Beltran AA, Smith JL, Drewry DH, Beltran AS, Axtman AD
Sci Rep. 13(1):6118. doi: 10.1038/s41598-023-32854-4
Publication date: April 14, 2023
PMID: 37059819
Davis-Gilbert ZW, Krämer A, Dunford JE, Howell S, Senbabaoglu F, Wells CI, Bashore FM, Havener TM, Smith JL, Hossain MA, Oppermann U, Drewry DH, Axtman AD
ACS Med Chem Lett. 14(4):432-441. doi: 10.1021/acsmedchemlett.2c00530
Publication date: April 13, 2023
PMID: 37077385
Dos Reis TF, de Castro PA, Bastos RW, Pinzan CF, Souza PFN, Ackloo S, Hossain MA, Drewry DH, Alkhazraji S, Ibrahim AS, Jo H, Lightfoot JD, Adams EM, Fuller KK, deGrado WF, Goldman GH
Nat Commun. 14(1):2052. doi: 10.1038/s41467-023-37573-y
Publication date: April 12, 2023
PMID: 37045836
Rak M, Tesch R, Berger LM, Shevchenko E, Raab M, Tjaden A, Zhubi R, Balourdas DI, Joerger AC, Poso A, Krämer A, Elson L, LuÄić A, Kronenberger T, Hanke T, Strebhardt K, Sanhaji M, Knapp S
Eur J Med Chem. 254:115347. doi: 10.1016/j.ejmech.2023.115347
Publication date: April 7, 2023
PMID: 37094449
Hanley RP, Nie DY, Tabor JR, Li F, Sobh A, Xu C, Barker NK, Dilworth D, Hajian T, Gibson E, Szewczyk MM, Brown PJ, Barsyte-Lovejoy D, Herring LE, Wang GG, Licht JD, Vedadi M, Arrowsmith CH, James LI
J Am Chem Soc. doi: 10.1021/jacs.3c01421
Publication date: March 28, 2023
PMID: 36976643
Yang X, Smith JL, Beck MT, Wilkinson JM, Michaud A, Vasta JD, Robers MB, Willson TM
Molecules. 28(7):. doi: 10.3390/molecules28072950
Publication date: March 25, 2023
PMID: 37049713
Li ASM, Kimani S, Wilson B, Noureldin M, González-Álvarez H, Mamai A, Hoffer L, Guilinger JP, Zhang Y, von Rechenberg M, Disch JS, Mulhern CJ, Slakman BL, Cuozzo JW, Dong A, Poda G, Mohammed M, Saraon P, Mittal M, Modh P, Rathod V, Patel B, Ackloo S, Santhakumar V, Szewczyk MM, Barsyte-Lovejoy D, Arrowsmith CH, Marcellus R, Guié MA, Keefe AD, Brown PJ, Halabelian L, Al-Awar R, Vedadi M
J Med Chem. doi: 10.1021/acs.jmedchem.2c02132
Publication date: March 22, 2023
PMID: 36948210
Tredup C, Ndreshkjana B, Schneider NS, Tjaden A, Kemas AM, Youhanna S, Lauschke VM, Berger BT, Krämer A, Berger LM, Röhm S, Knapp S, Farin HF, Müller S
ACS Chem Biol. doi: 10.1021/acschembio.2c00877
Publication date: March 21, 2023
PMID: 36944371
Dahlin JL, Hua BK, Zucconi BE, Nelson SD, Singh S, Carpenter AE, Shrimp JH, Lima-Fernandes E, Wawer MJ, Chung LPW, Agrawal A, O'Reilly M, Barsyte-Lovejoy D, Szewczyk M, Li F, Lak P, Cuellar M, Cole PA, Meier JL, Thomas T, Baell JB, Brown PJ, Walters MA, Clemons PA, Schreiber SL, Wagner BK
Nat Commun. 14(1):1364. doi: 10.1038/s41467-023-36829-x
Publication date: March 13, 2023
PMID: 36914634
Tang S, Garzon Sanz M, Smith O, Krämer A, Egbase D, Caton PW, Knapp S, Butterworth S
Acta Pharm Sin B. 13(2):709-721. doi: 10.1016/j.apsb.2022.07.016
Publication date: March 7, 2023
PMID: 36873168
Hasyeoui M, Lassagne F, Erb W, Nael M, Elokely KM, Chaikuad A, Knapp S, Jorda A, Vallés SL, Quissac E, Verreault M, Robert T, Bach S, Samarat A, Mongin F
Bioorg Chem. 134:106456. doi: 10.1016/j.bioorg.2023.106456
Publication date: March 4, 2023
PMID: 36913879
Aakula A, Sharma M, Tabaro F, Nätkin R, Kamila J, Honkanen H, Schapira M, Arrowsmith C, Nykter M, Westermarck J
Life Sci Alliance. 6(5):. doi: 10.26508/lsa.202301928
Publication date: March 2, 2023
PMID: 36858798
Arora R, Linders JTM, Aci-Sèche S, Verheyen T, Van Heerde E, Brehmer D, Chaikuad A, Knapp S, Bonnet P
Eur J Med Chem. 250:115231. doi: 10.1016/j.ejmech.2023.115231
Publication date: February 25, 2023
PMID: 36878151
Li ASM, Homsi C, Bonneil E, Thibault P, Verreault A, Vedadi M
Biochim Biophys Acta Gene Regul Mech. 194922. doi: 10.1016/j.bbagrm.2023.194922
Publication date: February 21, 2023
PMID: 36822575
Göricke F, Vu V, Smith L, Scheib U, Böhm R, Akkilic N, Wohlfahrt G, Weiske J, Bömer U, Brzezinka K, Lindner N, Lienau P, Gradl S, Beck H, Brown PJ, Santhakumar V, Vedadi M, Barsyte-Lovejoy D, Arrowsmith CH, Schmees N, Petersen K
J Med Chem. doi: 10.1021/acs.jmedchem.2c01933
Publication date: February 20, 2023
PMID: 36802665