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Gybeľ T, Čada Š, Klementová D, Schwalm MP, Berger BT, Šebesta M, Knapp S, Bryja V
J Biol Chem. 107407. doi: 10.1016/j.jbc.2024.107407
Publication date: May 23, 2024
PMID: 38796065
Chi G, Jaślan D, Kudrina V, Böck J, Li H, Pike ACW, Rautenberg S, Krogsaeter E, Bohstedt T, Wang D, McKinley G, Fernandez-Cid A, Mukhopadhyay SMM, Burgess-Brown NA, Keller M, Bracher F, Grimm C, Dürr KL
Structure. doi: 10.1016/j.str.2024.05.005
Publication date: May 23, 2024
PMID: 38815576
Owens DDG, Maitland MER, Khalili Yazdi A, Song X, Reber V, Schwalm MP, Machado RAC, Bauer N, Wang X, Szewczyk MM, Dong C, Dong A, Loppnau P, Calabrese MF, Dowling MS, Lee J, Montgomery JI, O'Connell TN, Subramanyam C, Wang F, Adamson EC, Schapira M, Gstaiger M, Knapp S, Vedadi M, Min J, Lajoie GA, Barsyte-Lovejoy D, Owen DR, Schild-Poulter C, Arrowsmith CH
Nat Chem Biol. doi: 10.1038/s41589-024-01618-0
Publication date: May 21, 2024
PMID: 38773330
Wellnitz J, Martin HJ, Anwar Hossain M, Rath M, Fox C, Popov KI, Willson TM, Muratov EN, Tropsha A
J Chem Inf Model. doi: 10.1021/acs.jcim.4c00412
Publication date: May 20, 2024
PMID: 38768560
Yong D, Ahmad S, Mabanglo MF, Halabelian L, Schapira M, Ackloo S, Perveen S, Ghiabi P, Vedadi M
Biochemistry. doi: 10.1021/acs.biochem.4c00044
Publication date: May 10, 2024
PMID: 38729622
Righetto GL, Yin Y, Duda DM, Vu V, Szewczyk MM, Zeng H, Li Y, Loppnau P, Mei T, Li YY, Seitova A, Patrick AN, Brazeau JF, Chaudhry C, Barsyte-Lovejoy D, Santhakumar V, Halabelian L
PNAS Nexus. 3(4):pgae153. doi: 10.1093/pnasnexus/pgae153
Publication date: April 26, 2024
PMID: 38665159
Schwalm MP, Saxena K, Müller S, Knapp S
Nat Protoc. doi: 10.1038/s41596-024-00979-z
Publication date: April 18, 2024
PMID: 38637703
Shah Zaib Saleem R, Schwalm MP, Knapp S
Bioorg Med Chem. 105:117718. doi: 10.1016/j.bmc.2024.117718
Publication date: April 12, 2024
PMID: 38621319
Schwarz M, Kurkunov M, Wittlinger F, Rudalska R, Wang G, Schwalm MP, Rasch A, Wagner B, Laufer SA, Knapp S, Dauch D, Gehringer M
J Med Chem. doi: 10.1021/acs.jmedchem.3c02483
Publication date: April 11, 2024
PMID: 38604131
Bedart C, Simoben CV, Schapira M
Curr Opin Struct Biol. 86:102812. doi: 10.1016/j.sbi.2024.102812
Publication date: April 10, 2024
PMID: 38603987
Eldeeb MA, Fallahi A, Soumbasis A, Bayne AN, Trempe JF, Fon EA
Autophagy. doi: 10.1080/15548627.2024.2340399
Publication date: April 10, 2024
PMID: 38597070
Champiré A, Berabez R, Braka A, Cosson A, Corret J, Girardin C, Serrano A, Aci-Sèche S, Bonnet P, Josselin B, Brindeau P, Ruchaud S, Leguevel R, Chatterjee D, Mathea S, Knapp S, Brion R, Verrecchia F, Vallée B, Plé K, Bénédetti H, Routier S
Eur J Med Chem. 271:116391. doi: 10.1016/j.ejmech.2024.116391
Publication date: April 9, 2024
PMID: 38669909
Asquith CRM, East MP, Laitinen T, Alamillo-Ferrer C, Hartikainen E, Wells CI, Axtman AD, Drewry DH, Tizzard GJ, Poso A, Willson TM, Johnson GL
Eur J Med Chem. 271:116357. doi: 10.1016/j.ejmech.2024.116357
Publication date: April 2, 2024
PMID: 38636130
Rasool S, Shomali T, Truong L, Croteau N, Veyron S, Bustillos BA, Springer W, Fiesel FC, Trempe JF
Sci Rep. 14(1):7739. doi: 10.1038/s41598-024-58285-3
Publication date: April 2, 2024
PMID: 38565869
Shen L, Ma X, Wang Y, Wang Z, Zhang Y, Pham HQH, Tao X, Cui Y, Wei J, Lin D, Abeywanada T, Hardikar S, Halabelian L, Smith N, Chen T, Barsyte-Lovejoy D, Qiu S, Xing Y, Yang Y
Nat Commun. 15(1):2809. doi: 10.1038/s41467-024-47107-9
Publication date: April 1, 2024
PMID: 38561334
Xiong Y, Greschik H, Johansson C, Seifert L, Gamble V, Park KS, Fagan V, Li F, Chau I, Vedadi M, Arrowsmith CH, Brennan P, Fedorov O, Jung M, Farnie G, Liu J, Oppermann U, Schüle R, Jin J
J Med Chem. doi: 10.1021/acs.jmedchem.4c00121
Publication date: March 27, 2024
PMID: 38533580
Yazdi AK, Perveen S, Dong C, Song X, Dong A, Szewczyk MM, Calabrese MF, Casimiro-Garcia A, Chakrapani S, Dowling MS, Ficici E, Lee J, Montgomery JI, O'Connell TN, Skrzypek GJ, Tran TP, Troutman MD, Wang F, Young JA, Min J, Barsyte-Lovejoy D, Brown PJ, Santhakumar V, Arrowsmith CH, Vedadi M, Owen DR
RSC Med Chem. 15(3):1066-1071. doi: 10.1039/d3md00633f
Publication date: March 20, 2024
PMID: 38516600
González-Álvarez H, Ensan D, Xin T, Wong JF, Zepeda-Velázquez CA, Cros J, Hoffer L, Kiyota T, Wilson BJ, Aman A, Roberts O, Isaac MB, Bullock AN, Smil D, Al-Awar R
J Med Chem. doi: 10.1021/acs.jmedchem.3c02308
Publication date: March 18, 2024
PMID: 38498998
Arrowsmith CH
Nat Struct Mol Biol. 31(3):395-396. doi: 10.1038/s41594-024-01244-3
Publication date: March 15, 2024
PMID: 38486110
Dötsch L, Davies C, Hennes E, Schönfeld J, Kumar A, Guita CDCL, Ehrler JHM, Hiesinger K, Thavam S, Janning P, Sievers S, Knapp S, Proschak E, Ziegler S, Waldmann H
J Med Chem. doi: 10.1021/acs.jmedchem.3c02245
Publication date: March 12, 2024
PMID: 38470246
Schapira M, Halabelian L, Arrowsmith CH, Harding RJ
Nat Chem Biol. doi: 10.1038/s41589-024-01570-z
Publication date: March 8, 2024
PMID: 38459278
Eldeeb MA, Bayne AN, Fallahi A, Goiran T, MacDougall EJ, Soumbasis A, Zorca CE, Tabah JJ, Thomas RA, Karpilovsky N, Mathur M, Durcan TM, Trempe JF, Fon EA
Proc Natl Acad Sci U S A. 121(10):e2313540121. doi: 10.1073/pnas.2313540121
Publication date: March 5, 2024
PMID: 38416681
Rak M, Menge A, Tesch R, Berger LM, Balourdas DI, Shevchenko E, Krämer A, Elson L, Berger BT, Abdi I, Wahl LM, Poso A, Kaiser A, Hanke T, Kronenberger T, Joerger AC, Müller S, Knapp S
J Med Chem. doi: 10.1021/acs.jmedchem.3c02217
Publication date: February 29, 2024
PMID: 38422480
Asressu KH, Smith JL, Dickmander RJ, Moorman NJ, Wellnitz J, Popov KI, Axtman AD, Willson TM
Pharmaceuticals (Basel). 17(3):. doi: 10.3390/ph17030306
Publication date: February 27, 2024
PMID: 38543092
Perveen S, Yazdi AK, Hajian T, Li F, Vedadi M
Sci Rep. 14(1):4509. doi: 10.1038/s41598-024-55184-5
Publication date: February 24, 2024
PMID: 38402266
Gilleran JA, Ashraf K, Delvillar M, Eck T, Fondekar R, Miller EB, Hutchinson A, Dong A, Seitova A, De Souza ML, Augeri D, Halabelian L, Siekierka J, Rotella DP, Gordon J, Childers WE, Grier MC, Staker BL, Roberge JY, Bhanot P
J Med Chem. doi: 10.1021/acs.jmedchem.3c01795
Publication date: February 19, 2024
PMID: 38372781
Gerninghaus J, Zhubi R, Kraemer A, Karim M, Tran DHN, Joerger AC, Schreiber C, Berger LM, Berger BT, Ehret TAL, Elson L, Lenz C, Saxena K, Mueller S, Einav S, Knapp S, Hanke T
bioRxiv. doi: 10.1101/2024.02.18.580805
Publication date: February 18, 2024
PMID: 38405908
Balzulat A, Zhu WF, Flauaus C, Hernandez-Olmos V, Heering J, Sethumadhavan S, Dubiel M, Frank A, Menge A, Hebchen M, Metzner K, Lu R, Lukowski R, Ruth P, Knapp S, Müller S, Steinhilber D, Hänelt I, Stark H, Proschak E, Schmidtko A
Adv Sci (Weinh). e2307237. doi: 10.1002/advs.202307237
Publication date: February 13, 2024
PMID: 38350720
Li F, Zhu WF, Empel C, Datsenko O, Kumar A, Xu Y, Ehrler JHM, Atodiresei I, Knapp S, Mykhailiuk PK, Proschak E, Koenigs RM
Science. 383(6682):498-503. doi: 10.1126/science.adm8095
Publication date: February 2, 2024
PMID: 38301027
Bauer N, Balourdas DI, Schneider JR, Zhang X, Berger LM, Berger BT, Schwalm MP, Klopp NA, Siveke JT, Knapp S, Joerger AC
ACS Chem Biol. doi: 10.1021/acschembio.3c00427
Publication date: January 31, 2024
PMID: 38291964
Xie SC, Wang Y, Morton CJ, Metcalfe RD, Dogovski C, Pasaje CFA, Dunn E, Luth MR, Kumpornsin K, Istvan ES, Park JS, Fairhurst KJ, Ketprasit N, Yeo T, Yildirim O, Bhebhe MN, Klug DM, Rutledge PJ, Godoy LC, Dey S, De Souza ML, Siqueira-Neto JL, Du Y, Puhalovich T, Amini M, Shami G, Loesbanluechai D, Nie S, Williamson N, Jana GP, Maity BC, Thomson P, Foley T, Tan DS, Niles JC, Han BW, Goldberg DE, Burrows J, Fidock DA, Lee MCS, Winzeler EA, Griffin MDW, Todd MH, Tilley L
Nat Commun. 15(1):937. doi: 10.1038/s41467-024-45224-z
Publication date: January 31, 2024
PMID: 38297033
Ipas H, Gouws EB, Abell NS, Chiou PC, Devanathan SK, Hervé S, Lee S, Mercado M, Reinsborough C, Halabelian L, Arrowsmith CH, Xhemalçe B
EMBO Rep. doi: 10.1038/s44319-024-00059-z
Publication date: January 23, 2024
PMID: 38263329
Mann MK, Wolf E, Silva M, Kwak HA, Wilson B, Bolotokova A, Wilson DJ, Harding RJ, Schapira M
ACS Omega. 9(1):917-924. doi: 10.1021/acsomega.3c07070
Publication date: January 9, 2024
PMID: 38222562
Galal KA, Krämer A, Strickland BG, Smith JL, Dickmander RJ, Moorman NJ, Willson TM
Bioorg Med Chem Lett. 99:129617. doi: 10.1016/j.bmcl.2024.129617
Publication date: January 8, 2024
PMID: 38199328
Rogov VV, Nezis IP, Tsapras P, Zhang H, Dagdas Y, Noda NN, Nakatogawa H, Wirth M, Mouilleron S, McEwan DG, Behrends C, Deretic V, Elazar Z, Tooze SA, Dikic I, Lamark T, Johansen T
Autophagy Rep. 2(1):. doi: 10.1080/27694127.2023.2188523
Publication date: December 31, 2023
PMID: 38214012
Amrhein JA, Berger LM, Balourdas DI, Joerger AC, Menge A, Krämer A, Frischkorn JM, Berger BT, Elson L, Kaiser A, Schubert-Zsilavecz M, Müller S, Knapp S, Hanke T
J Med Chem. doi: 10.1021/acs.jmedchem.3c01980
Publication date: December 21, 2023
PMID: 38126712
Takarada JE, Cunha MR, Almeida VM, Vasconcelos SNS, Santiago AS, Godoi PH, Salmazo A, Ramos PZ, Fala AM, de Souza LR, Da Silva IEP, Bengtson MH, Massirer KB, Couñago RM
Bioorg Med Chem. 98:117561. doi: 10.1016/j.bmc.2023.117561
Publication date: December 20, 2023
PMID: 38157838
Kimani SW, Perveen S, Szewezyk M, Zeng H, Dong A, Li F, Ghiabi P, Li Y, Chau I, Arrowsmith CH, Barsyte-Lovejoy D, Santhakumar V, Vedadi M, Halabelian L
Commun Biol. 6(1):1272. doi: 10.1038/s42003-023-05655-8
Publication date: December 16, 2023
PMID: 38104184
Ong HW, de Silva C, Avalani K, Kwarcinski F, Mansfield CR, Chirgwin M, Truong A, Derbyshire ER, Zutshi R, Drewry DH
ACS Med Chem Lett. 14(12):1774-1784. doi: 10.1021/acsmedchemlett.3c00354
Publication date: December 14, 2023
PMID: 38116430
Fnaiche A, Chan HC, Paquin A, González Suárez N, Vu V, Li F, Allali-Hassani A, Cao MA, Szewczyk MM, Bolotokova A, Allemand F, Gelin M, Barsyte-Lovejoy D, Santhakumar V, Vedadi M, Guichou JF, Annabi B, Gagnon A
ACS Med Chem Lett. 14(12):1746-1753. doi: 10.1021/acsmedchemlett.3c00386
Publication date: December 14, 2023
PMID: 38116405
Alqazzaz MA, Luciani GM, Vu V, Machado RAC, Szewczyk MM, Adamson EC, Cheon S, Li F, Arrowsmith CH, Minden MD, Barsyte-Lovejoy D
Exp Hematol. 104135. doi: 10.1016/j.exphem.2023.11.009
Publication date: December 10, 2023
PMID: 38072134
Lindberg MF, Deau E, Miege F, Greverie M, Roche D, George N, George P, Merlet L, Gavard J, Brugman SJT, Aret E, Tinnemans P, de Gelder R, Sadownik J, Verhofstad E, Sleegers D, Santangelo S, Dairou J, Fernandez-Blanco Ã, Dierssen M, Krämer A, Knapp S, Meijer L
J Med Chem. doi: 10.1021/acs.jmedchem.3c01888
Publication date: December 5, 2023
PMID: 38051674
Deng Y, Song X, Iyamu ID, Dong A, Min J, Huang R
Acta Pharm Sin B. 13(12):4893-4905. doi: 10.1016/j.apsb.2023.07.022
Publication date: December 4, 2023
PMID: 38045046
Outhwaite IR, Singh S, Berger BT, Knapp S, Chodera JD, Seeliger MA
Elife. 12:. doi: 10.7554/eLife.86189
Publication date: December 4, 2023
PMID: 38047771
Karelou M, Kampasis D, Kalampaliki AD, Persoons L, Krämer A, Schols D, Knapp S, De Jonghe S, Kostakis IK
Molecules. 28(23):. doi: 10.3390/molecules28237912
Publication date: December 2, 2023
PMID: 38067641
Sanz Murillo M, Villagran Suarez A, Dederer V, Chatterjee D, Alegrio Louro J, Knapp S, Mathea S, Leschziner AE
Sci Adv. 9(48):eadk6191. doi: 10.1126/sciadv.adk6191
Publication date: December 1, 2023
PMID: 38039358
Tiek D, Wells CI, Schröder M, Song X, Alamillo-Ferrer C, Goenka A, Iglesia R, Lu M, Hu B, Kwarcinski F, Sintha P, de Silva C, Hossain MA, Picado A, Zuercher W, Zutshi R, Knapp S, Riggins RB, Cheng SY, Drewry DH
Curr Res Chem Biol. 3:. doi: 10.1016/j.crchbi.2023.100045
Publication date: November 27, 2023
PMID: 38009092
Ahmad S, Xu J, Feng JA, Hutchinson A, Zeng H, Ghiabi P, Dong A, Centrella PA, Clark MA, Guié MA, Guilinger JP, Keefe AD, Zhang Y, Cerruti T, Cuozzo JW, von Rechenberg M, Bolotokova A, Li Y, Loppnau P, Seitova A, Li YY, Santhakumar V, Brown PJ, Ackloo S, Halabelian L
J Med Chem. doi: 10.1021/acs.jmedchem.3c01471
Publication date: November 23, 2023
PMID: 37996079
Ayoubi R, Ryan J, Biddle MS, Alshafie W, Fotouhi M, Bolivar SG, Ruiz Moleon V, Eckmann P, Worrall D, McDowell I, Southern K, Reintsch W, Durcan TM, Brown C, Bandrowski A, Virk H, Edwards AM, McPherson P, Laflamme C
Elife. 12:. doi: 10.7554/eLife.91645
Publication date: November 23, 2023
PMID: 37995198
Mende H, Khatri A, Lange C, Poveda-Cuevas SA, Tascher G, Covarrubias-Pinto A, Löhr F, Koschade SE, Dikic I, Münch C, Bremm A, Brunetti L, Brandts CH, Uckelmann H, Dötsch V, Rogov VV, Bhaskara RM, Müller S
Cell Rep. 42(12):113484. doi: 10.1016/j.celrep.2023.113484
Publication date: November 22, 2023
PMID: 37999976