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Scantlebury J, Vost L, Carbery A, Hadfield TE, Turnbull OM, Brown N, Chenthamarakshan V, Das P, Grosjean H, von Delft F, Deane CM
J Chem Inf Model. doi: 10.1021/acs.jcim.3c00322
Publication date: May 11, 2023
PMID: 37166179
Cunha MR, Catta-Preta CMC, Takarada JE, Moreira GA, Massirer KB, Couñago RM
J Biol Chem. 104807. doi: 10.1016/j.jbc.2023.104807
Publication date: May 10, 2023
PMID: 37172730
Durcan TM, Axtman AD
Front Cell Neurosci. 17:1196543. doi: 10.3389/fncel.2023.1196543
Publication date: May 1, 2023
PMID: 37124399
Hargittay B, Mineev KS, Richter C, Sreeramulu S, Jonker HRA, Saxena K, Schwalbe H
Biomol NMR Assign. doi: 10.1007/s12104-023-10132-8
Publication date: April 29, 2023
PMID: 37118562
Ong HW, Liang Y, Richardson W, Lowry ER, Wells CI, Chen X, Silvestre M, Dempster K, Silvaroli JA, Smith JL, Wichterle H, Pabla NS, Ultanir SK, Bullock AN, Drewry DH, Axtman AD
ACS Chem Neurosci. doi: 10.1021/acschemneuro.3c00135
Publication date: April 21, 2023
PMID: 37084253
Liu K, Zhang J, Xiao Y, Yang A, Song X, Li Y, Chen Y, Hughes TR, Min J
J Biol Chem. 104734. doi: 10.1016/j.jbc.2023.104734
Publication date: April 20, 2023
PMID: 37086783
Bashore FM, Marquez AB, Chaikuad A, Howell S, Dunn AS, Beltran AA, Smith JL, Drewry DH, Beltran AS, Axtman AD
Sci Rep. 13(1):6118. doi: 10.1038/s41598-023-32854-4
Publication date: April 14, 2023
PMID: 37059819
Davis-Gilbert ZW, Krämer A, Dunford JE, Howell S, Senbabaoglu F, Wells CI, Bashore FM, Havener TM, Smith JL, Hossain MA, Oppermann U, Drewry DH, Axtman AD
ACS Med Chem Lett. 14(4):432-441. doi: 10.1021/acsmedchemlett.2c00530
Publication date: April 13, 2023
PMID: 37077385
Dos Reis TF, de Castro PA, Bastos RW, Pinzan CF, Souza PFN, Ackloo S, Hossain MA, Drewry DH, Alkhazraji S, Ibrahim AS, Jo H, Lightfoot JD, Adams EM, Fuller KK, deGrado WF, Goldman GH
Nat Commun. 14(1):2052. doi: 10.1038/s41467-023-37573-y
Publication date: April 12, 2023
PMID: 37045836
Rak M, Tesch R, Berger LM, Shevchenko E, Raab M, Tjaden A, Zhubi R, Balourdas DI, Joerger AC, Poso A, Krämer A, Elson L, LuÄić A, Kronenberger T, Hanke T, Strebhardt K, Sanhaji M, Knapp S
Eur J Med Chem. 254:115347. doi: 10.1016/j.ejmech.2023.115347
Publication date: April 7, 2023
PMID: 37094449
Hanley RP, Nie DY, Tabor JR, Li F, Sobh A, Xu C, Barker NK, Dilworth D, Hajian T, Gibson E, Szewczyk MM, Brown PJ, Barsyte-Lovejoy D, Herring LE, Wang GG, Licht JD, Vedadi M, Arrowsmith CH, James LI
J Am Chem Soc. doi: 10.1021/jacs.3c01421
Publication date: March 28, 2023
PMID: 36976643
Yang X, Smith JL, Beck MT, Wilkinson JM, Michaud A, Vasta JD, Robers MB, Willson TM
Molecules. 28(7):. doi: 10.3390/molecules28072950
Publication date: March 25, 2023
PMID: 37049713
Li ASM, Kimani S, Wilson B, Noureldin M, González-Álvarez H, Mamai A, Hoffer L, Guilinger JP, Zhang Y, von Rechenberg M, Disch JS, Mulhern CJ, Slakman BL, Cuozzo JW, Dong A, Poda G, Mohammed M, Saraon P, Mittal M, Modh P, Rathod V, Patel B, Ackloo S, Santhakumar V, Szewczyk MM, Barsyte-Lovejoy D, Arrowsmith CH, Marcellus R, Guié MA, Keefe AD, Brown PJ, Halabelian L, Al-Awar R, Vedadi M
J Med Chem. doi: 10.1021/acs.jmedchem.2c02132
Publication date: March 22, 2023
PMID: 36948210
Tredup C, Ndreshkjana B, Schneider NS, Tjaden A, Kemas AM, Youhanna S, Lauschke VM, Berger BT, Krämer A, Berger LM, Röhm S, Knapp S, Farin HF, Müller S
ACS Chem Biol. doi: 10.1021/acschembio.2c00877
Publication date: March 21, 2023
PMID: 36944371
Dahlin JL, Hua BK, Zucconi BE, Nelson SD, Singh S, Carpenter AE, Shrimp JH, Lima-Fernandes E, Wawer MJ, Chung LPW, Agrawal A, O'Reilly M, Barsyte-Lovejoy D, Szewczyk M, Li F, Lak P, Cuellar M, Cole PA, Meier JL, Thomas T, Baell JB, Brown PJ, Walters MA, Clemons PA, Schreiber SL, Wagner BK
Nat Commun. 14(1):1364. doi: 10.1038/s41467-023-36829-x
Publication date: March 13, 2023
PMID: 36914634
Tang S, Garzon Sanz M, Smith O, Krämer A, Egbase D, Caton PW, Knapp S, Butterworth S
Acta Pharm Sin B. 13(2):709-721. doi: 10.1016/j.apsb.2022.07.016
Publication date: March 7, 2023
PMID: 36873168
Hasyeoui M, Lassagne F, Erb W, Nael M, Elokely KM, Chaikuad A, Knapp S, Jorda A, Vallés SL, Quissac E, Verreault M, Robert T, Bach S, Samarat A, Mongin F
Bioorg Chem. 134:106456. doi: 10.1016/j.bioorg.2023.106456
Publication date: March 4, 2023
PMID: 36913879
Aakula A, Sharma M, Tabaro F, Nätkin R, Kamila J, Honkanen H, Schapira M, Arrowsmith C, Nykter M, Westermarck J
Life Sci Alliance. 6(5):. doi: 10.26508/lsa.202301928
Publication date: March 2, 2023
PMID: 36858798
Arora R, Linders JTM, Aci-Sèche S, Verheyen T, Van Heerde E, Brehmer D, Chaikuad A, Knapp S, Bonnet P
Eur J Med Chem. 250:115231. doi: 10.1016/j.ejmech.2023.115231
Publication date: February 25, 2023
PMID: 36878151
Li ASM, Homsi C, Bonneil E, Thibault P, Verreault A, Vedadi M
Biochim Biophys Acta Gene Regul Mech. 194922. doi: 10.1016/j.bbagrm.2023.194922
Publication date: February 21, 2023
PMID: 36822575
Göricke F, Vu V, Smith L, Scheib U, Böhm R, Akkilic N, Wohlfahrt G, Weiske J, Bömer U, Brzezinka K, Lindner N, Lienau P, Gradl S, Beck H, Brown PJ, Santhakumar V, Vedadi M, Barsyte-Lovejoy D, Arrowsmith CH, Schmees N, Petersen K
J Med Chem. doi: 10.1021/acs.jmedchem.2c01933
Publication date: February 20, 2023
PMID: 36802665
Schuller M, Zarganes-Tzitzikas T, Bennett J, De Cesco S, Fearon D, von Delft F, Fedorov O, Brennan PE, Ahel I
Pathogens. 12(2):. doi: 10.3390/pathogens12020324
Publication date: February 15, 2023
PMID: 36839595
Schwalm MP, Knapp S, Rogov VV
J Cell Biochem. doi: 10.1002/jcb.30380
Publication date: February 13, 2023
PMID: 36780422
Li F, Ghiabi P, Hajian T, Klima M, Li ASM, Yazdi AK, Chau I, Loppnau P, Kutera M, Seitova A, Bolotokova A, Hutchinson A, Perveen S, Boura E, Vedadi M
Biochim Biophys Acta Gen Subj. 130319. doi: 10.1016/j.bbagen.2023.130319
Publication date: February 8, 2023
PMID: 36764586
MacDonald KM, Nicholson-Puthenveedu S, Tageldein MM, Khasnis S, Arrowsmith CH, Harding SM
Nat Commun. 14(1):556. doi: 10.1038/s41467-023-36195-8
Publication date: February 2, 2023
PMID: 36732527
Ali MM, Naz S, Ashraf S, Knapp S, Ul-Haq Z
Int J Biol Macromol. 123428. doi: 10.1016/j.ijbiomac.2023.123428
Publication date: January 26, 2023
PMID: 36709803
Barsyte-Lovejoy D
J Vis Exp. doi: 10.3791/64821
Publication date: January 20, 2023
PMID: 37602846
Denis HL, Alpaugh M, Alvarez CP, Fenyi A, Barker RA, Chouinard S, Arrowsmith CH, Melki R, Labib R, Harding RJ, Cicchetti F
Cell Mol Life Sci. 80(2):45. doi: 10.1007/s00018-023-04687-x
Publication date: January 18, 2023
PMID: 36651994
Outhwaite IR, Singh S, Berger BT, Knapp S, Chodera JD, Seeliger MA
bioRxiv. doi: 10.1101/2023.01.13.523972
Publication date: January 16, 2023
PMID: 36711619
Wells C, Liang Y, Pulliam TL, Lin C, Awad D, Eduful B, O'Byrne S, Hossain MA, Catta-Preta CMC, Ramos PZ, Gileadi O, Gileadi C, Couñago RM, Stork B, Langendorf CG, Nay K, Oakhill JS, Mukherjee D, Racioppi L, Means AR, York B, McDonnell DP, Scott JW, Frigo DE, Drewry DH
Cells. 12(2):. doi: 10.3390/cells12020287
Publication date: January 11, 2023
PMID: 36672221
Gahbauer S, Correy GJ, Schuller M, Ferla MP, Doruk YU, Rachman M, Wu T, Diolaiti M, Wang S, Neitz RJ, Fearon D, Radchenko DS, Moroz YS, Irwin JJ, Renslo AR, Taylor JC, Gestwicki JE, von Delft F, Ashworth A, Ahel I, Shoichet BK, Fraser JS
Proc Natl Acad Sci U S A. 120(2):e2212931120. doi: 10.1073/pnas.2212931120
Publication date: January 10, 2023
PMID: 36598939
Ong HW, Truong A, Kwarcinski F, de Silva C, Avalani K, Havener TM, Chirgwin M, Galal KA, Willis C, Krämer A, Liu S, Knapp S, Derbyshire ER, Zutshi R, Drewry DH
Eur J Med Chem. 249:115043. doi: 10.1016/j.ejmech.2022.115043
Publication date: December 30, 2022
PMID: 36736152
Balboa JR, Essig DJ, Ma S, Karer N, Clemmensen LS, Pedersen SW, Joerger AC, Knapp S, Østergaard S, Strømgaard K
J Med Chem. doi: 10.1021/acs.jmedchem.2c01803
Publication date: December 29, 2022
PMID: 36580549
Zhou J, Horton JR, Menna M, Fiorentino F, Ren R, Yu D, Hajian T, Vedadi M, Mazzoccanti G, Ciogli A, Weinhold E, Hüben M, Blumenthal RM, Zhang X, Mai A, Rotili D, Cheng X
J Med Chem. doi: 10.1021/acs.jmedchem.2c01789
Publication date: December 29, 2022
PMID: 36581322
Hogg DW, Reid AL, Dodsworth TL, Chen Y, Reid RM, Xu M, Husic M, Biga PR, Slee A, Buck LT, Barsyte-Lovejoy D, Locke M, Lovejoy DA
Front Physiol. 13:1031264. doi: 10.3389/fphys.2022.1031264
Publication date: December 17, 2022
PMID: 36523555
Tjaden A, Giessmann RT, Knapp S, Schröder M, Müller S
STAR Protoc. 3(4):101791. doi: 10.1016/j.xpro.2022.101791
Publication date: December 16, 2022
PMID: 36317177
Schröder M, Leiendecker M, Grädler U, Braun J, Blum A, Wanior M, Berger BT, Krämer A, Müller S, Esdar C, Knapp S, Heinrich T
J Med Chem. doi: 10.1021/acs.jmedchem.2c01705
Publication date: December 14, 2022
PMID: 36516476
Müller S, Frye S, Baell J
RSC Med Chem. 13(12):1438. doi: 10.1039/d2md90036j
Publication date: December 14, 2022
PMID: 36561071
Alshafie W, Fotouhi M, Shlaifer I, Ayoubi R, Edwards AM, Durcan TM, McPherson PS, Laflamme C
F1000Res. 11:977. doi: 10.12688/f1000research.124632.2
Publication date: December 7, 2022
PMID: 36415206
Hogg DW, Casatti CC, Belsham DD, Baršytė-Lovejoy D, Lovejoy DA
Biochem Biophys Rep. 32:101397. doi: 10.1016/j.bbrep.2022.101397
Publication date: December 6, 2022
PMID: 36467544
Preger C, Notarnicola A, Hellström C, Wigren E, Fernandes-Cerqueira C, Kvarnström M, Wahren-Herlenius M, Idborg H, Lundberg IE, Persson H, Gräslund S, Jakobsson PJ
J Autoimmun. 134:102951. doi: 10.1016/j.jaut.2022.102951
Publication date: December 2, 2022
PMID: 36470210
Ercoli MF, Ramos PZ, Jain R, Pilotte J, Dong OX, Thompson T, Wells CI, Elkins JM, Edwards AM, Couñago RM, Drewry DH, Ronald PC
Plant Direct. 6(11):e460. doi: 10.1002/pld3.460
Publication date: December 1, 2022
PMID: 36447653
Amrhein JA, Berger LM, Tjaden A, Krämer A, Elson L, Tolvanen T, Martinez-Molina D, Kaiser A, Schubert-Zsilavecz M, Müller S, Knapp S, Hanke T
Int J Mol Sci. 23(23):. doi: 10.3390/ijms232314834
Publication date: November 27, 2022
PMID: 36499165
Rovers E, Liu L, Schapira M
Comput Struct Biotechnol J. 20:6163-6171. doi: 10.1016/j.csbj.2022.11.010
Publication date: November 25, 2022
PMID: 36420167
Amrhein JA, Beyett TS, Feng WW, Krämer A, Weckesser J, Schaeffner IK, Rana JK, Jänne PA, Eck MJ, Knapp S, Hanke T
J Med Chem. doi: 10.1021/acs.jmedchem.2c01041
Publication date: November 16, 2022
PMID: 36384036
Stephenson Clarke JR, Douglas LR, Duriez PJ, Balourdas DI, Joerger AC, Khadiullina R, Bulatov E, Baud MGJ
ACS Pharmacol Transl Sci. 5(11):1169-1180. doi: 10.1021/acsptsci.2c00164
Publication date: November 11, 2022
PMID: 36407959
Chaikuad A, Zhubi R, Tredup C, Knapp S
IUCrJ. 9(Pt 6):720-727. doi: 10.1107/S2052252522008582
Publication date: November 1, 2022
PMID: 36381143
Payliss BJ, Tse YWE, Reichheld SE, Lemak A, Yun HY, Houliston S, Patel A, Arrowsmith CH, Sharpe S, Wyatt HDM
Cell Rep. 41(4):111537. doi: 10.1016/j.celrep.2022.111537
Publication date: October 25, 2022
PMID: 36288699
Antolin AA, Sanfelice D, Crisp A, Villasclaras Fernandez E, Mica IL, Chen Y, Collins I, Edwards A, Müller S, Al-Lazikani B, Workman P
Nucleic Acids Res. doi: 10.1093/nar/gkac909
Publication date: October 21, 2022
PMID: 36268860
Shell DJ, Rectenwald JM, Buttery PH, Johnson RL, Foley CA, Guduru SKR, Uguen M, Rubiano JS, Zhang X, Li F, Norris-Drouin JL, Axtman M, Brian Hardy P, Vedadi M, Frye SV, James LI, Pearce KH
SLAS Discov. doi: 10.1016/j.slasd.2022.10.003
Publication date: October 19, 2022
PMID: 36272689