Molecular insights into lipid-assisted Ca(2+) regulation of the TRP channel Polycystin-2. Read more about Molecular insights into lipid-assisted Ca(2+) regulation of the TRP channel Polycystin-2.
Insights into the RecQ helicase mechanism revealed by the structure of the helicase domain of human RECQL5. Read more about Insights into the RecQ helicase mechanism revealed by the structure of the helicase domain of human RECQL5.
The SUV4-20 inhibitor A-196 verifies a role for epigenetics in genomic integrity. Read more about The SUV4-20 inhibitor A-196 verifies a role for epigenetics in genomic integrity.
Development of potent, selective SRPK1 inhibitors as potential topical therapeutics for neovascular eye disease. Read more about Development of potent, selective SRPK1 inhibitors as potential topical therapeutics for neovascular eye disease.
Discovery of Potent and Selective Inhibitors for G9a-Like Protein (GLP) Lysine Methyltransferase. Read more about Discovery of Potent and Selective Inhibitors for G9a-Like Protein (GLP) Lysine Methyltransferase.
The EED protein-protein interaction inhibitor A-395 inactivates the PRC2 complex. Read more about The EED protein-protein interaction inhibitor A-395 inactivates the PRC2 complex.
Targeting human SET1/MLL family of proteins. Read more about Targeting human SET1/MLL family of proteins.
Discovery and structure activity relationship of the first potent cryptosporidium FIKK kinase inhibitor. Read more about Discovery and structure activity relationship of the first potent cryptosporidium FIKK kinase inhibitor.
Discovery of Peptidomimetic Ligands of EED as Allosteric Inhibitors of PRC2. Read more about Discovery of Peptidomimetic Ligands of EED as Allosteric Inhibitors of PRC2.
