Hinge Binder Scaffold Hopping Identifies Potent Calcium/Calmodulin-Dependent Protein Kinase Kinase 2 (CAMKK2) Inhibitor Chemotypes. Read more about Hinge Binder Scaffold Hopping Identifies Potent Calcium/Calmodulin-Dependent Protein Kinase Kinase 2 (CAMKK2) Inhibitor Chemotypes.
Histone and DNA binding ability studies of the NSD subfamily of PWWP domains. Read more about Histone and DNA binding ability studies of the NSD subfamily of PWWP domains.
A Concerted Action of UBA5 C-Terminal Unstructured Regions Is Important for Transfer of Activated UFM1 to UFC1. Read more about A Concerted Action of UBA5 C-Terminal Unstructured Regions Is Important for Transfer of Activated UFM1 to UFC1.
Crystal Structure-Guided Design of Bisubstrate Inhibitors and Photoluminescent Probes for Protein Kinases of the PIM Family. Read more about Crystal Structure-Guided Design of Bisubstrate Inhibitors and Photoluminescent Probes for Protein Kinases of the PIM Family.
Identification of Pyrimidine-Based Lead Compounds for Understudied Kinases Implicated in Driving Neurodegeneration. Read more about Identification of Pyrimidine-Based Lead Compounds for Understudied Kinases Implicated in Driving Neurodegeneration.
High-Throughput Crystallography Reveals Boron-Containing Inhibitors of a Penicillin-Binding Protein with Di- and Tricovalent Binding Modes. Read more about High-Throughput Crystallography Reveals Boron-Containing Inhibitors of a Penicillin-Binding Protein with Di- and Tricovalent Binding Modes.
Production of Recombinant PRMT Proteins using the Baculovirus Expression Vector System. Read more about Production of Recombinant PRMT Proteins using the Baculovirus Expression Vector System.
Discovery and Characterization of Selective and Ligand-Efficient DYRK Inhibitors. Read more about Discovery and Characterization of Selective and Ligand-Efficient DYRK Inhibitors.
Trends in kinase drug discovery: targets, indications and inhibitor design. Read more about Trends in kinase drug discovery: targets, indications and inhibitor design.
