Assessing reversible and irreversible binding effects of kinase covalent inhibitors through ADP-Glo assays. Read more about Assessing reversible and irreversible binding effects of kinase covalent inhibitors through ADP-Glo assays.
Quantitative Methods to Study Protein Arginine Methyltransferase 1-9 Activity in Cells. Read more about Quantitative Methods to Study Protein Arginine Methyltransferase 1-9 Activity in Cells.
Structural and functional characterization of ubiquitin variant inhibitors for the JAMM-family deubiquitinases STAMBP and STAMBPL1. Read more about Structural and functional characterization of ubiquitin variant inhibitors for the JAMM-family deubiquitinases STAMBP and STAMBPL1.
Structure and Function of Protein Arginine Methyltransferase PRMT7. Read more about Structure and Function of Protein Arginine Methyltransferase PRMT7.
Non-canonical role of Hippo tumor suppressor serine/threonine kinase 3 STK3 in prostate cancer. Read more about Non-canonical role of Hippo tumor suppressor serine/threonine kinase 3 STK3 in prostate cancer.
Discovery of a Potent Dual SLK/STK10 Inhibitor Based on a Maleimide Scaffold. Read more about Discovery of a Potent Dual SLK/STK10 Inhibitor Based on a Maleimide Scaffold.
A NSD3-targeted PROTAC suppresses NSD3 and cMyc oncogenic nodes in cancer cells. Read more about A NSD3-targeted PROTAC suppresses NSD3 and cMyc oncogenic nodes in cancer cells.
Development of a Selective Dual Discoidin Domain Receptor (DDR)/p38 Kinase Chemical Probe. Read more about Development of a Selective Dual Discoidin Domain Receptor (DDR)/p38 Kinase Chemical Probe.
Novel quaternary structures of the human prion protein globular domain. Read more about Novel quaternary structures of the human prion protein globular domain.
Design and Development of a Chemical Probe for Pseudokinase Ca2+/calmodulin-Dependent Ser/Thr Kinase. Read more about Design and Development of a Chemical Probe for Pseudokinase Ca2+/calmodulin-Dependent Ser/Thr Kinase.
