Synthesis and biological evaluation of Haspin inhibitors: Kinase inhibitory potency and cellular activity. Read more about Synthesis and biological evaluation of Haspin inhibitors: Kinase inhibitory potency and cellular activity.
A Consensus Compound/Bioactivity Dataset for Data-Driven Drug Design and Chemogenomics. Read more about A Consensus Compound/Bioactivity Dataset for Data-Driven Drug Design and Chemogenomics.
AD Informer Set: Chemical tools to facilitate Alzheimer's disease drug discovery. Read more about AD Informer Set: Chemical tools to facilitate Alzheimer's disease drug discovery.
Protein proximity networks and functional evaluation of the Casein Kinase 1 γ family reveal unique roles for CK1γ3 in WNT signaling. Read more about Protein proximity networks and functional evaluation of the Casein Kinase 1 γ family reveal unique roles for CK1γ3 in WNT signaling.
Enabling pseudokinases as potential drug targets. Read more about Enabling pseudokinases as potential drug targets.
Calcium/calmodulin-dependent protein kinase kinase 2 regulates hepatic fuel metabolism. Read more about Calcium/calmodulin-dependent protein kinase kinase 2 regulates hepatic fuel metabolism.
PRMT inhibition induces a viral mimicry response in triple-negative breast cancer. Read more about PRMT inhibition induces a viral mimicry response in triple-negative breast cancer.
Illuminating the Dark: Highly Selective Inhibition of Serine/Threonine Kinase 17A with Pyrazolo[1,5-a]pyrimidine-Based Macrocycles. Read more about Illuminating the Dark: Highly Selective Inhibition of Serine/Threonine Kinase 17A with Pyrazolo[1,5-a]pyrimidine-Based Macrocycles.
Structure and activity of human TMPRSS2 protease implicated in SARS-CoV-2 activation. Read more about Structure and activity of human TMPRSS2 protease implicated in SARS-CoV-2 activation.
