Ribosomal oxygenases are structurally conserved from prokaryotes to humans. Read more about Ribosomal oxygenases are structurally conserved from prokaryotes to humans.
A Series of Potent CREBBP Bromodomain Ligands Reveals an Induced-Fit Pocket Stabilized by a Cation-π Interaction. Read more about A Series of Potent CREBBP Bromodomain Ligands Reveals an Induced-Fit Pocket Stabilized by a Cation-π Interaction.
Structural basis for histone mimicry and hijacking of host proteins by influenza virus protein NS1. Read more about Structural basis for histone mimicry and hijacking of host proteins by influenza virus protein NS1.
Multiparameter Optimization in CNS Drug Discovery: Design of Pyrimido[4,5-d]azepines as Potent 5-Hydroxytryptamine 2C (5-HT2C) Receptor Agonists with Exquisite Functional Selectivity over 5-HT2A and 5-HT2B Receptors. Read more about Multiparameter Optimization in CNS Drug Discovery: Design of Pyrimido[4,5-d]azepines as Potent 5-Hydroxytryptamine 2C (5-HT2C) Receptor Agonists with Exquisite Functional Selectivity over 5-HT2A and 5-HT2B Receptors.
Synthesis, Optimization, and Evaluation of Novel Small Molecules as Antagonists of WDR5-MLL Interaction. Read more about Synthesis, Optimization, and Evaluation of Novel Small Molecules as Antagonists of WDR5-MLL Interaction.
Discovery and development of potent and selective inhibitors of histone methyltransferase g9a. Read more about Discovery and development of potent and selective inhibitors of histone methyltransferase g9a.
A comparison of protein kinases inhibitor screening methods using both enzymatic activity and binding affinity determination. Read more about A comparison of protein kinases inhibitor screening methods using both enzymatic activity and binding affinity determination.
STRUCTURAL CHARACTERIZATION OF HUMAN CHOLESTEROL 7α-HYDROXYLASE. Read more about STRUCTURAL CHARACTERIZATION OF HUMAN CHOLESTEROL 7α-HYDROXYLASE.
Linking genotypes database with locus-specific database and genotype-phenotype correlation in phenylketonuria. Read more about Linking genotypes database with locus-specific database and genotype-phenotype correlation in phenylketonuria.
Discovery and Optimization of Small-Molecule Ligands for the CBP/p300 Bromodomains. Read more about Discovery and Optimization of Small-Molecule Ligands for the CBP/p300 Bromodomains.
