SGC chemical probes are open-access reagents that are meant to be used by the biomedical research community with no restrictions on use. SGC-developed probes are complemented by a growing set of donated high-quality chemical probes developed in industry and non-SGC laboratories. These are also available for unencumbered use.
The table below contains the entire collection of probes from SGC’s chemical probes program and donated chemical probes. To browse the collection, find associated data, or acquire samples, select the desired chemical probe in the table below and follow the links that appear on that page. You can sort the table by clicking the column headers.
For inquiries or requests related to chemical probes or libraries, please contact us at proberequests@thesgc.org.
Name | Structures | Protein Family | Target Protein | Negative Control | Cellular usage | Added |
---|---|---|---|---|---|---|
JNJ-8003 |
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RNA polymerase | RSV-L | JNJ-6643 | ||
JNJ-78911118 |
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Glutamate-gated ion channel | GRIN2A | JNJ-77914993 | up to 10 µM | |
ACBI3 |
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GTPase | KRAS | cis-ACBI3 | 1-10 µM | |
THNAN69 |
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Kinase | LIMK2 | THNAN69-NC | 10 -100 nM | |
SM311 |
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Kinase | LIMK1 | SM311-NC | 0.1 - 1 µM | |
BI-5121 |
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GPCR | HCRTR1 | BI-6199 | 100 nM | |
BAY-439 |
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Phospholipase A2 | PLA2G5 | BAY-163 | up to 300 nM | |
SGC-NSP2hel-1 |
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Helicases | CHIKV_nsp2 helicase | SGC-NSP2hel-1N | 1 µM | |
JYQ-173 |
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Peptidase C56 | PARK7 | MB078 | Up to 1 µM | |
Huib32 |
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Deubiquitinase | USP32 | Huib32NC | 5 µM | |
JNJ-79883960 |
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Receptor | NRLP3 | JNJ-78832000 | up to 10 µM | |
SGC-NSP2PRO-1 |
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Protease | CHIKV_nsp2 | SGC-NSP2PRO-1N | ||
LH168 |
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WD40 repeat | WDR5 | LH222 | 1 µM | |
OICR-41103 |
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WD40 repeat | DCAF1 | OICR-41103N | 1 µM; not to exceed 5 µM | |
BI-1915 |
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Protease | CTSS | BI-1920 | 1 µM | |
BI-113823 |
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GPCR | BDKRB1 | BI-5832 | 100 nM | |
JNJ-54082730 |
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Hydrolase | PDE2A | JNJ-54103985 | 1 µM | |
JNJ-3738 |
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Kinase | CDK7 | JNJ-6240 | 1 µM | |
BAY-9835 |
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Protease | ADAMTS7, ADAMTS12 | BAY-1880 | 100 nM | |
SGC-CDKL2/AAK1/BMP2K-1 |
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Kinase | CDKL2 | CDKL2/AAK1/BMP2K -1N | ≤1 µM | |
ABT-724 |
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GPCR | DRD4 | A-769 | ||
BAY-474 |
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Kinase | MET | BAY-827 | ||
BAY-7598 |
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Protease | MMP12 | BAY-694 | ||
BI 99179 |
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Synthase | FASN | BI 99990 | ||
ERKi |
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Kinase | MAPK3, MAPK1 | ERKi-NC | ||
(R)-9s |
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GPCR | ADRA1D | (S)-9s | ||
A-485 |
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Transferase | EP300, CREBBP | A-486 | ||
ABT-100 |
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Transferase | FNTB | A-108 | ||
BAY-386 |
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GPCR | F2R | BAY-448 | ||
BAY-707 |
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Hydrolase | NUDT1 | BAY-604 | ||
BI-1935 |
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Hydrolase | EPHX2 | BI-2049 | ||
BI-9627 |
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Solute carriers | SLC9A1 | BI-0054 | ||
BTZO-1 |
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Cytokine | MIF | BTZO-4 | ||
CRTH2 antagonist |
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GPCR | PTGDR2 | CRTH2 negative control | ||
GSM1 |
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Protease | Gamma secretase complex | GSM-NC | ||
MRK-560 |
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Protease | Gamma secretase complex | GSI-NC | ||
MRL-650 |
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GPCR | CNR1 | MRL-CB1-NC | ||
MRL-SYKi |
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Kinase | SYK | MRL-SYKi-NC | ||
PF-04418948 |
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GPCR | PTGER2 | PF-04475866 | ||
PF-05105679 |
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Ion channel | TRPM8 | PF-05257137 | ||
TP-004 |
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Protease | METAP2 | TPn-004 | ||
A-079 |
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Ion channel | TRPA1 | A-226 | ||
ABT-546 |
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GPCR | EDNRA | A-545 | ||
BAY-1797 |
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Ion channel | P2X4 | BAY-207 | ||
BAY-678 |
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Protease | ELANE | BAY-677 | ||
BAY-784 |
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GPCR | GNRHR | BAY-786 | ||
BAY-876 |
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Solute carriers | SLC2A1 | BAY-588 | ||
BAY-885 |
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Kinase | MAPK7 | BAY-693 | ||
BI 639667 |
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GPCR | CCR1 | BI-9307 | ||
BI 653048 |
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Nuclear hormone receptor | NR3C1 | BI-3047 | ||
BI-1950 |
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Integrin | ITGAL | BI-9446 | ||
BI-2545 |
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Phosphodiesterase | ENPP2 | BI-3017 | ||
BI-4394 |
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Protease | MMP13 | BI-4395 | ||
KISS1-305 |
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GPCR | KISS1R | KISS1-543 | ||
PF-04457845 |
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Hydrolase | FAAH | PF-04875474 | ||
T-26c |
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Protease | MMP13 | T-26f | ||
TP-020 |
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Transferase | MGAT2 | TP-020n | ||
TP-021 |
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Transcription factor | BCL6 | TP-021n | ||
A-1155463 |
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Regulator protein | BCL2L1 | A-1107969 | ||
A-1211212 |
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Regulator protein | BCL2 | A-1210227 | ||
A-1596586 |
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Ion channel | CFTR | A-1596584 | ||
A-192621 |
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GPCR | EDNRB | A-1806262 | ||
BAY-293 |
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Nucleotide exchange factor | SOS1 | BAY-294 | ||
BAY-549 |
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Kinase | ROCK1, ROCK2 | BAY-4900 | ||
BI-1230 |
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Protease | HCV NS3 | BI-1675 | ||
IPP/CNRS-A017 |
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Dehydrogenase | DHODH | IPP/CNRS-A019 | ||
MLi-2 |
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Kinase | LRRK2 | MLi-2-NC | ||
MSD-CYP11B2 |
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Cytochrome P450 | CYP11B2 | MSD-CYP11B2 Negative control | ||
MSD-M1PAM |
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GPCR | CHRM1 | MSD-M1PAM-NC | ||
PPTN |
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GPCR | P2RY14 | PPTN-NC | ||
T3-CLK |
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Kinase | CLK1, CLK2, CLK3, CLK4 | T3-CLK-N | ||
THPP-1 |
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Phosphodiesterase | PDE10A | THPP-1-NC | ||
TP-008 |
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Kinase | ACVR1B, TGFBR1 | Al11 | ||
TP-024 |
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GPCR | GPR52 | TP-024n | ||
UCSF924 |
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GPCR | DRD4 | UCSF924NC | ||
(R)-ZINC-3573 |
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GPCR | MRGPRX2 | (S)-ZINC-3573 | ||
BAY-069 |
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Amino acid transaminase | BCAT1, BCAT2 | BAY-771 | ||
BAY-179 |
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Protease | Complex I | BAY-070 | Yes | |
BAY-3827 |
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Kinase | PRKAA1, RPS6KA1 | BAY-974 | ||
BAY-390 |
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Ion channel | TRPA1 | BAY-9897 | ||
BAY-899 |
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GPCR | LHCGR | BAY-897 | ||
BAY-985 |
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Kinase | TBK1, IKBKE | BAY-440 | ||
BI-2540 |
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Reverse transcriptase | HIV NNRT | BI-2439 | ||
FS-694 |
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Kinase | MAPK14 | FM-743 | ||
NVS-MALT1 |
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Protease | MALT1 | NVS-MALT1-C | ||
Ogerin |
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GPCR | GPR68 | ZINC32547799 | ||
Skepinone-L |
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Kinase | MAPK14 | FM-743 | ||
SR-302 |
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Kinase | DDR1, DDR2, MAPK11, MAPK14 | SR-301 | ||
SR-318 |
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Kinase | MAPK14 | SR-321 | ||
TP-030-1 |
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Kinase | RIPK1 | TP-030n | ||
TP-030-2 |
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Kinase | RIPK1 | TP-030n | ||
WM-1119 |
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Transferase | KAT6A, KAT6B | WM-2474 | ||
8RK64 |
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Regulator protein | UCHL1 | JYQ88 | ||
A-446 |
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Hydrolase | GLS | A-426 | ||
BAY-091 |
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Kinase | PIP4K2A | BAY-0361 | ||
BAY-3153 |
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GPCR | CCR1 | BAY-173 | ||
BAY-6672 |
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GPCR | PTGFR | BAY-403 | ||
BI 207127 |
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RNA polymerase | HCV NS5B | BI-7656 | ||
BI 605906 |
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Kinase | IKBKB | BI-5026 | ||
BI-1942 | Protease | CMA1 | ||||
Borussertib |
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Kinase | AKT1, AKT2 | RL2578 | ||
GSK046 | Bromodomains | BRD2, BRD3, BRD4, BRDT | ||||
GSK620 | Bromodomains | BRD2, BRD3, BRD4, BRDT | ||||
GSK778 | Bromodomains | BRD2, BRD3, BRD4, BRDT | ||||
GSK789 |
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Bromodomains | BRD2, BRD3, BRD4, BRDT | GSK791 | ||
GSK973 |
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Bromodomains | BRD2, BRD3, BRD4, BRDT | GSK943 | ||
JNJ-42396302 | Phosphodiesterase | PDE10A | JNJ-40573663 | |||
JNJ-54119936 |
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Nuclear hormone receptor | RORC | JNJ-53721590 | ||
MSC-4381 |
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Monocarboxylate transporter | SLC16A3 | MSC-0516 | ||
PFI-653 |
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Hydrolase | VNN1 | PFI-653-N | ||
TP-040 |
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Hydrolase | OGA | TP-040n | ||
BAY 1816032 |
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Kinase | BUB1 | BAY-283 | ||
BAY1125976 |
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Kinase | AKT1/2 | BAY-940 | ||
BI-2081 |
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GPCR | FFAR1 | BI-0340 | ||
CCT369260 |
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Transcription factor | BCL6 | CCT393732 | ||
GNE-2256 |
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Kinase | IRAK4 | GNE-6689 | ||
JNJ-39758979 |
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GPCR | HRH4 | JNJ-39668551 | ||
JNJ-6204 |
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Kinase | CSNK1D/CSNK1E | JNJ-0293 | ||
JNJ-65355394 |
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Hydrolase | OGA | JNJ-73924149 | ||
JNJ-9350 |
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Oxidase | SMOX | JNJ-4545 | ||
SAFit2 |
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Isomerase | FKBP5 | ddSAFit2 | ||
TP-050 |
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Ion channel | GRIN2A | TP-050n | ||
TP-051 |
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GPCR | FFAR1 | TP-051n | ||
TP-061 |
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Helicases | Brr2 | TP-061N | 5 µM | |
SGC-UBD1031 |
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UBD (ubiquitin binding domain) | USP16/HDAC6 | SGC-UBD1031N | 10 µM | |
BAY 1816032 |
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2OG | BUB1 | BAY-283 | ||
OICR11029 |
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Transcription factor | BCL6 | OICR11600 | 1 µM | |
PFI-8 |
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YEATS | YEATS | PFI-8N | 1 µM | |
UNC8732 |
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Methyl Lysine Binder | NSD2 | UNC8884 | 3 µM | |
BAY-277 |
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Aminopeptidase | METAP2 | BAY-8805 | ||
BI-5524 |
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Chymotrypsin | ELANE | BI-5525 | ||
BIBO3304 |
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GPCR | NPY1R | BIBO3457 | ||
SGK3-PROTAC1 |
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Kinase | SGK3 | cisSGK3-PROTAC1 | ||
VZ185 |
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Bromodomain-containing protein family | BRD7, BRD9 | cisVZ185 | ||
WEB2086 |
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GPCR | PTAFR | WEB2387 | ||
BAY 1753011 |
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GPCR | AVPR1A, AVPR2 | BAY-2297 | ||
BAY-6096 |
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GPCR | ADRA2B | BAY-726 | ||
JA310 |
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Kinase | MST3, MST4 | JA262 | < 1 µM | |
BI-3802 |
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Transcription factor | BCL6 | BI-5273 | ||
BI-3812 |
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Transcription factor | BCL6 | BI-5273 | ||
BI-8668 |
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Sodium channels | Epithelial sodium channel (ENaC) | BI-0337 | ||
JP3000 |
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Nuclear hormone receptor | RXRA, RXRB, RXRG | JP3001 | ||
SGC-CAF382-1 |
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Kinase | CDKL5 | SGC-CAF268-1N | ≤ 100 nM | |
SGC-CDKL5/GSK3 |
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Kinase | CDKL5, GSK3 | SGC-CDKL5/GSK3-1N | 100 nM | |
SGC-GSK3-1 |
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Kinase | GSK3 | SGC-CDKL5/GSK3-1N | 100 nM | |
BAY-7081 |
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Phoshodiesterase | PDE9A | BAY-7424 | ||
JNJ-42226314 |
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Serine hydrolase | MGLL | JNJ-8034 | ||
JNJ-4355 |
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BCL2 protein family | MCL1 | JNJ-78732576 | ||
TP-060 |
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Glucosyltransferase | UGCG | TP-060n | ||
BI-3231 |
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17β-hydroxysteroid dehydrogenases | HSD17B13 | BI-0955 | ||
FHT-2344 |
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SWI/SNF | SMARCA2, SMARCA4 | FHT-5908 | ||
TH-257 |
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Kinase | LIMK1, LIMK2 | TH-263 | 1 µM | |
JA397 |
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Kinase | CDK14-18 | JA314 | < 1 µM | |
SGC-CK2-2 |
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Kinase | CK2/CSNK2 | SGK-CK2-2N | 1 µM | |
SGC-PI5P4Kγ/MYLK4-1 |
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Kinase | PI5P4K gamma, MYLK4 | SGC-PI5P4Kγ/MYLK4-1N | 100 nM | |
LIJTF500025 |
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Kinase | LIMK1, LIMK2 | LIJTF500120 | < 1 µM | |
CS640 |
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Kinase | CAMK1 | CS640s | < 1 µM | |
MSC1186 |
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Kinase | SRPK | MSC5360 | < 1 µM | |
BAY-805 |
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USP (ubiquitin specific protease) | USP21 | BAY-728 | 1 µM | |
MRK-952 |
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Hydrolase | NUDT5 | MRK-952-NC | < 1 µM | |
MRK-990 |
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Methyltransferase | PRMT9, PRMT5 | MRK-990-NC | < 10 µM | |
MU1742 |
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Kinase | CK1delta, CK1epsilon | MU2027 | 1 µM | |
SGC-PIKFYVE-1 |
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Kinase | PIKfyve | SGC-PIKFYVE-1N | 100 nM | |
M4K2234 |
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Kinase | ALK1, ALK2 | M4K2234NC | 1 µM | |
MU1700 |
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Kinase | ALK1, ALK2 | MU1700NC | 1 µM | |
SGC-UBD253 |
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UBD (ubiquitin binding domain) | HDAC6 | SGC-UBD253N | 3 µM | |
CK156 |
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Kinase | STK17A, DRAK1 | CKJB71 | 5 µM | |
PFI-7 |
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E3 ligase | GID4 | PFI-7N | 1 µM | |
MRIA9 |
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Kinase | SIK1, SIK2, SIK3 | MR7 | 10 µM | |
Homer |
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WD40 repeat | WDR5 | nc_WDR5, nc_VHL | 1 µM | |
SGC-SMARCA-BRDVIII |
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Bromodomains | PB1(5), SMARCA2/4 | SGC-BRDVIII-NC | 10 µM | |
NR162 |
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Kinase | CASK | NR187 | 10 µM | |
PFI-6 |
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YEATS | MLLT1, MLLT3 | PFI-6N | 1 µM | |
SGC-CK2-1 |
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Kinase | CSNK2A1, CSNK2A2 | SGC-CK2-1N | 100 nM | |
NVS-MLLT-1 |
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YEATS | MLLT1, MLLT3 | NVS-MLLT-C | 1 µM | |
SGC-CLK-1 |
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Kinase | CLK1, CLK2, CLK4 | SGC-CLK-1N | 1 µM | |
SGC-STK17B-1 |
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Kinase | STK17B, DRAK2 | SGC-STK17B-1N | 1 µM | |
SGC-CAMKK2-1 |
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Kinase | CAMKK1, CAMKK2 | SGC-CAMKK2-1N | 1 µM | |
PFI-5 |
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Methyltransferase | SMYD2 | PFI-5N | 1 µM | |
SGC6870 |
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Methyltransferase | PRMT6 | SGC6870N | 1 µM | |
UNC6934 |
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Methyl Lysine Binder | NSD2-PWWP1 | UNC7145 | 1 µM | |
MU1210 |
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Kinase | CLK1, CLK2, CLK4, DYRK1A, DYRK1B, DYRK2 | MU140 | 1 µM | |
NVS-BPTF-1 |
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Bromodomains | BPTF | NVS-BPTF-C | < 1 µM | |
TP-238 |
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Bromodomains | CECR2, BPTF | TP-422 | < 2 µM | |
VinSpinIn |
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Spindlin domains | Spin1 | VinSpinIC | 0.5 µM - 3 µM | |
DDR-TRK-1 |
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Kinase | DDR, TRK | DDR-TRK-1N | 5 µM | |
SKI-73 |
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Methyltransferase | CARM1 | SKI-73N | 1 µM | |
BI-9321 |
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Methyl Lysine Binder | NSD3 | BI-9466 | 0.5 µM - 20 µM | |
MRK-740 |
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Methyltransferase | PRDM9 | MRK-740-NC | 3 µM | |
BAY-826 |
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Kinase | TIE1, TEK, DDR1, DDR2 | BAY-309 | ||
BI-665915 |
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Lipoxygenase | ALOX5AP | BI-0153 | ||
SGC3027 |
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Methyltransferase | PRMT7 | SGC3027N | 1 µM | |
SGC-AAK1-1 |
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Kinase | AAK1, BMP2K, BIKE | SGC-AAK1-1N | 1 µM | |
SGC-GAK-1 |
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Kinase | GAK | SGC-GAK-1N | 1 µM | |
BI01383298 |
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Solute carriers | SLC13A5 | BI01372674 | 1 µM | |
L-Moses |
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Bromodomains | KAT2A, KAT2B | D-Moses | 1 µM | |
BAY-6035 |
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Methyltransferase | SMYD3 | BAY-444 | 1 µM | |
GSK4027 |
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Bromodomains | KAT2A, KAT2B | GSK4028 | 1 µM | |
FM-381 |
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Kinase | JAK3 | FM-479 | 100 nM | |
BAY-850 |
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Bromodomains | ATAD2 | BAY-460 | 1 µM | |
GSK6853 |
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Bromodomains | BRPF1 | GSK9311 | < 1 µM | |
GSK8814 |
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Bromodomains | ATAD2, ATAD2B | GSK8815 | 1 µM | |
A-395 |
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WD40 repeat | EED | A-395N | 100 nM | |
LLY-283 |
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Methyltransferase | PRMT5 | LLY-284 | 1 µM | |
NVS-PAK1-1 |
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Kinase | PAK1 | NVS-PAK1-C | 1 µM | |
BAY-299 |
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Bromodomains | TAF1, BRD1 | BAY-364 | 1 µM | |
TP-064 |
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Methyltransferase | CARM1 | TP-064N | 1 µM | |
TP-472 |
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Bromodomains | BRD9, BRD7 | TP-472N | 1 µM | |
GSK864 |
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Dehydrogenase | IDH1 | GSK990 | 1 µM | |
MS023 |
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Methyltransferase | PRMT1, PRMT3, CARM1, PRMT6, PRMT8 | MS094 | 1 µM | |
A-196 |
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Methyltransferase | SUV420H1, SUV420H2 | SGC2043 | 1 µM | |
GSK591 |
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Methyltransferase | PRMT5 | SGC2096 | 1 µM | |
MS049 |
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Methyltransferase | CARM1, PRMT6 | MS049N | 1 µM | |
NVS-CECR2-1 |
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Bromodomains | CECR2 | NVS-CECR2-C | 1 µM | |
I-BRD9 |
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Bromodomains | BRD9 | 1 µM | ||
BAY-598 |
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Methyltransferase | SMYD2 | BAY-369 | 1 µM | |
BI-9564 |
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Bromodomains | BRD9, BRD7 | 1 µM | ||
GSK484 |
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Arginine deiminases | PAD4 | GSK106 | 1 µM | |
GSK2801 |
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Bromodomains | BAZ2A, BAZ2B | GSK8573 | 1 µM | |
LP99 |
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Bromodomains | BRD9, BRD7 | 2S,3R-enantiomer | 1 µM | |
NI-57 |
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Bromodomains | BRPF1, BRD1, BRPF3 | 1 µM | ||
PFI-4 |
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Bromodomains | BRPF1 | 1 µM | ||
OF-1 |
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Bromodomains | BRPF1, BRD1, BRPF3 | <5 µM | ||
SGC707 |
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Methyltransferase | PRMT3 | XY1 | 1 µM | |
BAZ2-ICR |
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Bromodomains | BAZ2A, BAZ2B | 1 µM | ||
OICR-9429 |
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WD40 repeat | WDR5 | OICR-0547 | 1 µM | |
GSK-LSD1 |
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Lysine Demethylase | KDM1A/LSD1 | 100 nM | ||
LLY-507 (multiple off-targets) |
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Methyltransferase | SMYD2 | SGC705 | 1 µM | |
PFI-3 |
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Bromodomains | SMARCA2, PBRM1, SMARCA4 | PFI-3oMet | 1 µM | |
A-366 |
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Methyltransferase | EHMT1/GLP, EHMT2/G9a | 1 µM | ||
(R)-PFI-2 |
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Methyltransferase | SETD7 | (S)-PFI-2 | 1 µM | |
UNC1999 |
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Methyltransferase | EZH2 | UNC2400 | 1 µM | |
I-CBP112 |
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Bromodomains | CREBBP, EP300 | 1 µM | ||
SGC-CBP30 |
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Bromodomains | CREBBP, EP300 | BDOIA513 | 1 µM | |
Bromosporine (BSP) |
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Bromodomains | pan-Bromodomain | 5 µM | ||
GSK343 |
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Methyltransferase | EZH2 | 1 µM | ||
UNC0642 |
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Methyltransferase | EHMT2/G9a, EHMT1/GLP | 1 µM | ||
UNC1215 |
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Methyl Lysine Binder | L3MBTL3 | UNC1079 | 1 µM | |
GSK-J1 |
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Lysine Demethylase | KDM6B/JMJD3, KDM6A/UTX, KDM5B/JARID1B | GSK-J2 (GSK-J5) | 100 nM | |
SGC0946 |
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Methyltransferase | DOT1L | SGC0649 | 1 µM | |
IOX2 |
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2OG | PHD2 | 1 µM | ||
IOX1 |
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2OG | Pan-KDM | 1 µM - 20 µM | ||
PFI-1 |
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Bromodomains | BRD2, BRD3, BRD4, BRDT | 1 µM | ||
(+)-JQ1 |
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Bromodomains | BRD2, BRD3, BRD4, BRDT | (-)-JQ1 | 1 µM | |
UNC0638 |
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Methyltransferase | EHMT2/G9a, EHMT1/GLP | UNC0737 | ≤ 1 µM |